Wednesday, July 8, 2026

Drug profile · INN

dolutegravir sodium

dolutegravir sodium (TIVICAY) is a human immunodeficiency virus type 1 integrase inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved PMDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — dolutegravir sodium
US status
approved
Class
Route
ORAL
Patents
0
Programs
0
Data quality
0.84

Quick answer

dolutegravir sodium (TIVICAY) is a human immunodeficiency virus type 1 integrase inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN dolutegravir sodium
Brand TIVICAY
Mechanism Human immunodeficiency virus type 1 integrase inhibitor
Target Human immunodeficiency virus type 1 integrase
Route ORAL
Formulation TABLET, FOR SUSPENSION

Mechanism of action

Human immunodeficiency virus type 1 integrase inhibitor

Primary target: Human immunodeficiency virus type 1 integrase

Approval history

Authority Status Date
FDA approved
PMDA approved

Related & competitor drugs

  1. bictegravir sodium Human immunodeficiency virus type 1 integrase inhibitor
  2. cabotegravir Antiinfectives for systemic use (J05)
  3. cabotegravir sodium Human immunodeficiency virus type 1 integrase inhibitor
  4. elvitegravir Antiinfectives for systemic use (J05)
  5. raltegravir potassium Antiinfectives for systemic use (J05)
  6. bictegravir Antiinfectives for systemic use (J05)

Frequently asked questions

What is dolutegravir sodium?

dolutegravir sodium (TIVICAY) is a human immunodeficiency virus type 1 integrase inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for dolutegravir sodium?

TIVICAY is a marketed brand name for dolutegravir sodium. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of dolutegravir sodium?

dolutegravir sodium has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.