Wednesday, July 8, 2026

Drug profile · INN

bictegravir sodium

bictegravir sodium (BIKTARVY) is a human immunodeficiency virus type 1 integrase inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 9
Pipeline programs 1
News articles 2
Drug details — bictegravir sodium

Quick answer

bictegravir sodium (BIKTARVY) is a human immunodeficiency virus type 1 integrase inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN bictegravir sodium
Brand BIKTARVY
Mechanism Human immunodeficiency virus type 1 integrase inhibitor
Target Human immunodeficiency virus type 1 integrase
Route ORAL
Formulation TABLET

Mechanism of action

Human immunodeficiency virus type 1 integrase inhibitor

Primary target: Human immunodeficiency virus type 1 integrase

Approval history

Authority Status Date
FDA approved

Recent coverage

Pipeline programs

  1. AT-01B-006 Phase 1 · Atea Pharmaceuticals · Healthy Volunteer Study

Related & competitor drugs

  1. cabotegravir Antiinfectives for systemic use (J05)
  2. cabotegravir sodium Human immunodeficiency virus type 1 integrase inhibitor
  3. dolutegravir sodium Human immunodeficiency virus type 1 integrase inhibitor
  4. elvitegravir Antiinfectives for systemic use (J05)
  5. raltegravir potassium Antiinfectives for systemic use (J05)
  6. bictegravir Antiinfectives for systemic use (J05)

Related patents

  1. US 12226429

    Highly active compounds against COVID-19

    Expires Mon Feb 13 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 11813278

    Highly active compounds against COVID-19

    Expires Mon Nov 09 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 11738038

    Highly active compounds against COVID-19

    Expires Mon Aug 24 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 11707480

    Highly active compounds against COVID-19

    Expires Mon Jul 20 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 10888529

    Vehicles for the transfection of miRNAs

    Expires Mon Jan 07 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 10874687

    Highly active compounds against COVID-19

    Expires Mon Dec 24 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. US 10610597

    Polycarbonates bearing aromatic N-heterocycles for drug delivery

    Expires Mon Apr 02 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. US 9919027

    Lipid nanoparticle of polymyxin

    Expires Mon Mar 15 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. US 9717797

    Polycarbonates bearing aromatic N-heterocycles for drug delivery

    Expires Mon Jul 27 2037 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is bictegravir sodium?

bictegravir sodium (BIKTARVY) is a human immunodeficiency virus type 1 integrase inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for bictegravir sodium?

BIKTARVY is a marketed brand name for bictegravir sodium. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of bictegravir sodium?

bictegravir sodium has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.