Saturday, July 11, 2026

Drug profile · INN

ciclosporin

ciclosporin (APO-CICLOSPORIN) is a cyclophilin a modulator. Associated with Novartis Pharmaceuticals.

EMA: approved TGA: approved Sensory organs (S01) S01XA18
Patents linked 0
Pipeline programs 10
News articles 0
Drug details — ciclosporin
Class
Sensory organs (S01)
Route
Patents
0
Programs
10
Data quality
0.83

Quick answer

ciclosporin (APO-CICLOSPORIN) is a cyclophilin a modulator. Associated with Novartis Pharmaceuticals.

Key facts

INN ciclosporin
Brand APO-CICLOSPORIN
Mechanism Cyclophilin A modulator
Target Peptidyl-prolyl cis-trans isomerase A
Therapeutic class Sensory organs (S01)
ATC code S01XA18

Mechanism of action

Cyclophilin A modulator

Primary target: Peptidyl-prolyl cis-trans isomerase A

Approval history

Authority Status Date
EMA approved
TGA approved

Pipeline programs

  1. KYV101-006 Phase 3 · Kyverna Therapeutics · Generalized myasthenia gravis
  2. Liposomal Ciclosporin A, Liposomal Ciclosporin A Phase 3 · ZAMBON S.P.A · Bronchiolitis Obliterans Syndrome in Patients post Single or
  3. CMAS825D12201 Phase 2 · Novartis India · Autoinflammatory diseases including NLRC4-Gain of Function (
  4. Ciclosporin Phase 2 · United Therapeutics Europe · Myocardial Reperfusion Injury
  5. P120142 Phase 2 · PARItec · Patient with newly diagnosed (≤ 3 months) type 1 diabetes st
  6. Verkazia 1 mg/mL eye drops, emulsion Phase 2 · HRA Pharma · Vernal Keratoconjunctivitis (VKC)
  7. 54659 Approved · Disc Medicine · Hand eczema
  8. Prednisolone Soluble Tablets for kidney transplant Approved · Disc Medicine · kidney transplant

Related & competitor drugs

  1. aflibercept Sensory organs (S01)
  2. atropine sulfate Sensory organs (S01)
  3. bimatoprost Sensory organs (S01)
  4. cyclosporine Cyclophilin A modulator
  5. atropine Sensory organs (S01)
  6. brinzolamide Sensory organs (S01)

Frequently asked questions

What is ciclosporin?

ciclosporin (APO-CICLOSPORIN) is a cyclophilin a modulator. Associated with Novartis Pharmaceuticals.

What is the brand name for ciclosporin?

APO-CICLOSPORIN is a marketed brand name for ciclosporin. Check FDA Drugs@FDA for the current US label holder and prescribing information.