Wednesday, July 8, 2026

Drug profile · INN

azilsartan kamedoxomil

azilsartan kamedoxomil (AZILSARTAN MEDOXOMIL AND CHLORTHALIDONE) is a type-1 angiotensin ii receptor antagonist. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 3
Pipeline programs 17
News articles 0
Drug details — azilsartan kamedoxomil
US status
approved
Class
Route
ORAL
Patents
3
Programs
17
Data quality
0.84

Quick answer

azilsartan kamedoxomil (AZILSARTAN MEDOXOMIL AND CHLORTHALIDONE) is a type-1 angiotensin ii receptor antagonist. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN azilsartan kamedoxomil
Brand AZILSARTAN MEDOXOMIL AND CHLORTHALIDONE
Mechanism Type-1 angiotensin II receptor antagonist
Target Type-1 angiotensin II receptor
Route ORAL
Formulation TABLET

Mechanism of action

Type-1 angiotensin II receptor antagonist

Primary target: Type-1 angiotensin II receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Azilsartan Phase 3 · Takeda · Pediatric Hypertension
  2. Azilsartan Medoxomil Phase 3 · Takeda · Hypertension
  3. Azilsartan Medoxomil and amlodipine Phase 3 · Takeda · Hypertension
  4. Azilsartan medoxomil and chlorthalidone Phase 3 · Takeda · Safety
  5. Azilsartan medoxomil and chlorthalidone Phase 3 · Takeda · Hypertension
  6. Azilsartan medoxomil and chlorthalidone Phase 3 · Takeda · Essential Hypertension
  7. Azilsartan medoxomil and olmesartan Phase 3 · Takeda · Hypertension
  8. Azilsartan medoxomil with or without add-on chlorthalidone Phase 3 · Takeda · Hypertension

Related & competitor drugs

  1. candesartan cilexetil Type-1 angiotensin II receptor antagonist
  2. irbesartan Cardiovascular system (C09)
  3. losartan potassium Type-1 angiotensin II receptor antagonist
  4. olmesartan medoxomil Type-1 angiotensin II receptor antagonist
  5. telmisartan Cardiovascular system (C09)
  6. valsartan Type-1 angiotensin II receptor antagonist

Related patents

  1. US 9387249

    Methods of treating hypertension with at least one angiotensin II receptor blocker and chlorthalidone

    Expires Mon Jul 07 2036 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 9169238

    Solid pharmaceutical composition

    Expires Mon Oct 22 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 9066936

    Solid pharmaceutical composition comprising a benzimidazole-7-carboxylate derivative and a pH control agent

    Expires Mon Jun 25 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is azilsartan kamedoxomil?

azilsartan kamedoxomil (AZILSARTAN MEDOXOMIL AND CHLORTHALIDONE) is a type-1 angiotensin ii receptor antagonist. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for azilsartan kamedoxomil?

AZILSARTAN MEDOXOMIL AND CHLORTHALIDONE is a marketed brand name for azilsartan kamedoxomil. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of azilsartan kamedoxomil?

azilsartan kamedoxomil has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.