Wednesday, July 8, 2026

Drug profile · INN

olmesartan medoxomil

olmesartan medoxomil (BENICAR) is a type-1 angiotensin ii receptor antagonist. Associated with Amneal Pharma Europe Ltd. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 2
News articles 0
Drug details — olmesartan medoxomil
US status
approved
Class
Route
ORAL
Patents
0
Programs
2
Data quality
0.89

Quick answer

olmesartan medoxomil (BENICAR) is a type-1 angiotensin ii receptor antagonist. Associated with Amneal Pharma Europe Ltd. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN olmesartan medoxomil
Brand BENICAR
Mechanism Type-1 angiotensin II receptor antagonist
Target Type-1 angiotensin II receptor
Route ORAL
Formulation TABLET

Mechanism of action

Type-1 angiotensin II receptor antagonist

Primary target: Type-1 angiotensin II receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. CXXB750A12201 Phase 2 · Novartis India · Heart Failure
  2. olmesartan medoxomil Phase 2 · Daiichi Sankyo US · Chronic Glomerulonephritis

Related & competitor drugs

  1. candesartan cilexetil Type-1 angiotensin II receptor antagonist
  2. irbesartan Cardiovascular system (C09)
  3. losartan potassium Type-1 angiotensin II receptor antagonist
  4. telmisartan Cardiovascular system (C09)
  5. valsartan Type-1 angiotensin II receptor antagonist
  6. angiotensin ii acetate Type-1 angiotensin II receptor agonist

Frequently asked questions

What is olmesartan medoxomil?

olmesartan medoxomil (BENICAR) is a type-1 angiotensin ii receptor antagonist. Associated with Amneal Pharma Europe Ltd. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for olmesartan medoxomil?

BENICAR is a marketed brand name for olmesartan medoxomil. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of olmesartan medoxomil?

olmesartan medoxomil has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.