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First People's Hospital

First People's Hospital drug portfolio — 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

SAN DIEGO, CA, CN HQ
NMPA registrant Type
Company details
Status
Public
HQ
SAN DIEGO, CA, CN
Programs
1136
Drugs
626
Patents
123
Intelligence · Drug Pipeline

First People's Hospital pipeline

Portfolio lens on 200 drugs and development assets — regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

First People's Hospital drug portfolio — 200 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

200 compounds
  1. abacavir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved.

  2. abatacept

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: T-lymphocyte activation antigen CD80.

    Target
    T-lymphocyte activation antigen CD80
    Mechanism
    T-lymphocyte activation antigen CD80 inhibitor
  3. US regulatory status: approved. Molecular target: Synaptosomal-associated protein 25.

    Target
    Synaptosomal-associated protein 25
    Mechanism
    Synaptosomal-associated protein 25 inhibitor
  4. acalabrutinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  5. US regulatory status: approved. Molecular target: Tyrosine-protein kinase BTK.

    Target
    Tyrosine-protein kinase BTK
    Mechanism
    Tyrosine-protein kinase BTK inhibitor
  6. US regulatory status: approved. Molecular target: Fatty-acid amide hydrolase 1.

    Target
    Fatty-acid amide hydrolase 1
    Mechanism
    Cyclooxygenase inhibitor
  7. US regulatory status: approved. Molecular target: Carbonic anhydrase 1.

    Target
    Carbonic anhydrase 1
    Mechanism
    Carbonic anhydrase XII inhibitor
  8. US regulatory status: approved. Mechanism: Glutathione precursor.

    Mechanism
    Glutathione precursor
  9. US regulatory status: approved. Molecular target: Retinoid receptor.

    Target
    Retinoid receptor
    Mechanism
    Retinoid receptor agonist
  10. US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  11. US regulatory status: approved. Molecular target: DNA polymerase catalytic subunit.

    Target
    DNA polymerase catalytic subunit
    Mechanism
    Human herpesvirus 1 DNA polymerase inhibitor
  12. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  13. Development asset linked to First People's Hospital in public FDA and regional records.

  14. Development asset linked to First People's Hospital in public FDA and regional records.

  15. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Adrenergic receptor.

    Target
    Adrenergic receptor
    Mechanism
    Adrenergic receptor agonist
  16. aflibercept

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Placenta growth factor.

    Target
    Placenta growth factor
    Mechanism
    Placenta growth factor inhibitor
  17. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Cytotoxic T-lymphocyte protein 4.

    Target
    Cytotoxic T-lymphocyte protein 4
    Mechanism
    Cytotoxic T-lymphocyte protein 4 inhibitor
  18. ala

    Development asset linked to First People's Hospital in public FDA and regional records.

  19. Development asset linked to First People's Hospital in public FDA and regional records.

  20. Development asset linked to First People's Hospital in public FDA and regional records.

  21. US regulatory status: approved. Molecular target: Beta-2 adrenergic receptor.

    Target
    Beta-2 adrenergic receptor
    Mechanism
    Beta-2 adrenergic receptor agonist
  22. US regulatory status: approved.

  23. US regulatory status: approved. Molecular target: Interleukin-2 receptor.

    Target
    Interleukin-2 receptor
    Mechanism
    Interleukin-2 receptor agonist
  24. alirocumab

    Cardiovascular system (C10)

    US regulatory status: approved. Molecular target: Proprotein convertase subtilisin/kexin type 9.

    Target
    Proprotein convertase subtilisin/kexin type 9
    Mechanism
    Subtilisin/kexin type 9 inhibitor
  25. Development asset linked to First People's Hospital in public FDA and regional records.

  26. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  27. alogliptin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Mechanism: Dipeptidyl peptidase IV inhibitor.

    Mechanism
    Dipeptidyl peptidase IV inhibitor
  28. US regulatory status: approved. Molecular target: Prostaglandin E2 receptor EP1 subtype.

    Target
    Prostaglandin E2 receptor EP1 subtype
    Mechanism
    Prostanoid EP1 receptor agonist
  29. US regulatory status: approved. Molecular target: Tissue-type plasminogen activator.

    Target
    Tissue-type plasminogen activator
    Mechanism
    Tissue-type plasminogen activator exogenous protein
  30. US regulatory status: approved. Mechanism: Antacid.

    Mechanism
    Antacid
  31. Development asset linked to First People's Hospital in public FDA and regional records.

  32. ambrisentan

    Cardiovascular system (C02)

    US regulatory status: approved. Molecular target: Endothelin receptor, ET-A/ET-B.

    Target
    Endothelin receptor, ET-A/ET-B
    Mechanism
    Endothelin receptor, ET-A/ET-B antagonist
  33. amikacin

    Antiinfectives for systemic use (J01)

    Antiinfectives for systemic use (J01) compound in First People's Hospital's portfolio.

  34. Development asset linked to First People's Hospital in public FDA and regional records. Mechanism: Serotonin transporter inhibitor.

    Mechanism
    Serotonin transporter inhibitor
  35. US regulatory status: approved. Molecular target: Sodium-dependent noradrenaline transporter.

    Target
    Sodium-dependent noradrenaline transporter
    Mechanism
    Norepinephrine transporter inhibitor
  36. amlodipine

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in First People's Hospital's portfolio. Mechanism: Voltage-gated L-type calcium channel blocker.

    Mechanism
    Voltage-gated L-type calcium channel blocker
  37. US regulatory status: approved. Molecular target: Voltage-gated L-type calcium channel.

    Target
    Voltage-gated L-type calcium channel
    Mechanism
    Voltage-gated L-type calcium channel blocker
  38. US regulatory status: approved. Molecular target: Voltage-gated L-type calcium channel.

    Target
    Voltage-gated L-type calcium channel
    Mechanism
    Voltage-gated L-type calcium channel blocker
  39. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  40. Development asset linked to First People's Hospital in public FDA and regional records.

  41. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Platelet-derived growth factor receptor beta.

    Target
    Platelet-derived growth factor receptor beta
    Mechanism
    Platelet-derived growth factor receptor beta inhibitor
  42. Development asset linked to First People's Hospital in public FDA and regional records.

  43. Various (V09) compound in First People's Hospital's portfolio. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  44. Development asset linked to First People's Hospital in public FDA and regional records.

  45. Development asset linked to First People's Hospital in public FDA and regional records.

  46. Development asset linked to First People's Hospital in public FDA and regional records.

  47. Development asset linked to First People's Hospital in public FDA and regional records.

  48. Development asset linked to First People's Hospital in public FDA and regional records.

  49. aprepitant

    Alimentary tract and metabolism (A04)

    US regulatory status: approved. Molecular target: Substance-P receptor.

    Target
    Substance-P receptor
    Mechanism
    Neurokinin 1 receptor antagonist
  50. US regulatory status: approved. Molecular target: Prothrombin.

    Target
    Prothrombin
    Mechanism
    Thrombin inhibitor
  51. Development asset linked to First People's Hospital in public FDA and regional records.

  52. asenapine

    Nervous system (N05)

    US regulatory status: approved. Mechanism: Serotonin 2a (5-HT2a) receptor antagonist.

    Mechanism
    Serotonin 2a (5-HT2a) receptor antagonist
  53. Development asset linked to First People's Hospital in public FDA and regional records.

  54. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  55. Development asset linked to First People's Hospital in public FDA and regional records. Mechanism: HMG-CoA reductase inhibitor.

    Mechanism
    HMG-CoA reductase inhibitor
  56. US regulatory status: approved. Molecular target: 3-hydroxy-3-methylglutaryl-coenzyme A reductase.

    Target
    3-hydroxy-3-methylglutaryl-coenzyme A reductase
    Mechanism
    HMG-CoA reductase inhibitor
  57. Development asset linked to First People's Hospital in public FDA and regional records.

  58. atropine sulfate

    Sensory organs (S01)

    US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M1.

    Target
    Muscarinic acetylcholine receptor M1
    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  59. aumolertinib

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in First People's Hospital's portfolio. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  60. Development asset linked to First People's Hospital in public FDA and regional records.

  61. Development asset linked to First People's Hospital in public FDA and regional records.

  62. avapritinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Platelet-derived growth factor receptor alpha.

    Target
    Platelet-derived growth factor receptor alpha
    Mechanism
    Stem cell growth factor receptor inhibitor
  63. azacitidine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 3A inhibitor
  64. azathioprine

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Amidophosphoribosyltransferase.

    Target
    Amidophosphoribosyltransferase
    Mechanism
    Amidophosphoribosyltransferase inhibitor
  65. US regulatory status: approved. Molecular target: Amidophosphoribosyltransferase.

    Target
    Amidophosphoribosyltransferase
    Mechanism
    Amidophosphoribosyltransferase inhibitor
  66. US regulatory status: approved. Molecular target: GABA-B receptor.

    Target
    GABA-B receptor
    Mechanism
    GABA-B receptor agonist
  67. US regulatory status: approved. Mechanism: Diagnostic agent.

    Mechanism
    Diagnostic agent
  68. basiliximab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Interleukin-2 receptor.

    Target
    Interleukin-2 receptor
    Mechanism
    Interleukin-2 receptor inhibitor
  69. Development asset linked to First People's Hospital in public FDA and regional records.

  70. Development asset linked to First People's Hospital in public FDA and regional records.

  71. bedaquiline

    Antiinfectives for systemic use (J04)

    Antiinfectives for systemic use (J04) compound in First People's Hospital's portfolio.

  72. Development asset linked to First People's Hospital in public FDA and regional records.

  73. bevacizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Vascular endothelial growth factor A, long form.

    Target
    Vascular endothelial growth factor A, long form
    Mechanism
    Vascular endothelial growth factor A inhibitor
  74. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Hepatitis C virus serine protease, NS3/NS4A.

    Target
    Hepatitis C virus serine protease, NS3/NS4A
    Mechanism
    Hepatitis C virus serine protease, NS3/NS4A inhibitor
  75. Development asset linked to First People's Hospital in public FDA and regional records.

  76. Development asset linked to First People's Hospital in public FDA and regional records. Mechanism: Probiotic.

    Mechanism
    Probiotic
  77. Development asset linked to First People's Hospital in public FDA and regional records.

  78. Development asset linked to First People's Hospital in public FDA and regional records.

  79. bivalirudin

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Prothrombin.

    Target
    Prothrombin
    Mechanism
    Thrombin inhibitor
  80. Development asset linked to First People's Hospital in public FDA and regional records.

  81. blinatumomab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: B-lymphocyte antigen CD19.

    Target
    B-lymphocyte antigen CD19
    Mechanism
    T cell surface glycoprotein CD3 cross-linking agent
  82. botulinum toxin type a

    Musculo-skeletal system (M03)

    Musculo-skeletal system (M03) compound in First People's Hospital's portfolio. Molecular target: Synaptosomal-associated protein 25.

    Target
    Synaptosomal-associated protein 25
    Mechanism
    Synaptosomal nerve-associated protein 25 (SNAP-25) hydrolytic enzyme
  83. Development asset linked to First People's Hospital in public FDA and regional records.

  84. brentuximab vedotin

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  85. budesonide

    Alimentary tract and metabolism (A07)

    US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  86. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  87. bupivacaine

    Nervous system (N01)

    US regulatory status: approved. Molecular target: Sodium channel protein type 4 subunit alpha.

    Target
    Sodium channel protein type 4 subunit alpha
    Mechanism
    Sodium channel protein type IV alpha subunit blocker
  88. US regulatory status: approved. Molecular target: Sodium channel protein type 4 subunit alpha.

    Target
    Sodium channel protein type 4 subunit alpha
    Mechanism
    Sodium channel protein type IV alpha subunit blocker
  89. US regulatory status: approved. Molecular target: 5-hydroxytryptamine receptor 1A.

    Target
    5-hydroxytryptamine receptor 1A
    Mechanism
    Serotonin 1a (5-HT1a) receptor partial agonist
  90. busulfan

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  91. Development asset linked to First People's Hospital in public FDA and regional records.

  92. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Cytotoxic T-lymphocyte protein 4.

    Target
    Cytotoxic T-lymphocyte protein 4
    Mechanism
    Cytotoxic T-lymphocyte protein 4 inhibitor
  93. US regulatory status: approved. Molecular target: Vitamin D3 receptor.

    Target
    Vitamin D3 receptor
    Mechanism
    Vitamin D receptor agonist
  94. US regulatory status: approved.

  95. US regulatory status: approved. Mechanism: Dihydrofolate reductase inhibitor.

    Mechanism
    Dihydrofolate reductase inhibitor
  96. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 antagonist
  97. canagliflozin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Sodium/glucose cotransporter 2.

    Target
    Sodium/glucose cotransporter 2
    Mechanism
    Sodium/glucose cotransporter 2 inhibitor
  98. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  99. Development asset linked to First People's Hospital in public FDA and regional records.

  100. Development asset linked to First People's Hospital in public FDA and regional records.

  101. US regulatory status: approved. Molecular target: Angiotensin-converting enzyme.

    Target
    Angiotensin-converting enzyme
    Mechanism
    Angiotensin-converting enzyme inhibitor
  102. Development asset linked to First People's Hospital in public FDA and regional records.

  103. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  104. carfilzomib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: 26S proteasome.

    Target
    26S proteasome
    Mechanism
    26S proteosome inhibitor
  105. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  106. Development asset linked to First People's Hospital in public FDA and regional records.

  107. US regulatory status: approved. Molecular target: Bacterial penicillin-binding protein.

    Target
    Bacterial penicillin-binding protein
    Mechanism
    Bacterial penicillin-binding protein inhibitor
  108. celecoxib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Prostaglandin G/H synthase 2.

    Target
    Prostaglandin G/H synthase 2
    Mechanism
    Cyclooxygenase-2 inhibitor
  109. Development asset linked to First People's Hospital in public FDA and regional records.

  110. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  111. cetuximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  112. Development asset linked to First People's Hospital in public FDA and regional records.

  113. Development asset linked to First People's Hospital in public FDA and regional records.

  114. Development asset linked to First People's Hospital in public FDA and regional records.

  115. Development asset linked to First People's Hospital in public FDA and regional records.

  116. US regulatory status: approved. Molecular target: Solute carrier family 12 member 3.

    Target
    Solute carrier family 12 member 3
    Mechanism
    Thiazide-sensitive sodium-chloride cotransporter inhibitor
  117. US regulatory status: approved. Molecular target: Estrogen receptor beta.

    Target
    Estrogen receptor beta
    Mechanism
    Estrogen receptor beta modulator
  118. US regulatory status: approved. Molecular target: Bile acids.

    Target
    Bile acids
    Mechanism
    Bile acids sequestering agent
  119. cholic acid

    Alimentary tract and metabolism (A05)

    US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  120. Development asset linked to First People's Hospital in public FDA and regional records.

  121. ciclosporin

    Sensory organs (S01)

    Sensory organs (S01) compound in First People's Hospital's portfolio. Molecular target: Peptidyl-prolyl cis-trans isomerase A.

    Target
    Peptidyl-prolyl cis-trans isomerase A
    Mechanism
    Cyclophilin A modulator
  122. US regulatory status: approved. Molecular target: cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A.

    Target
    cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
    Mechanism
    Phosphodiesterase 3A inhibitor
  123. US regulatory status: approved. Molecular target: Bacterial DNA gyrase.

    Target
    Bacterial DNA gyrase
    Mechanism
    Bacterial DNA gyrase inhibitor
  124. US regulatory status: approved. Molecular target: Bacterial DNA gyrase.

    Target
    Bacterial DNA gyrase
    Mechanism
    Bacterial DNA gyrase inhibitor
  125. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  126. Development asset linked to First People's Hospital in public FDA and regional records. Mechanism: Serotonin transporter inhibitor.

    Mechanism
    Serotonin transporter inhibitor
  127. Development asset linked to First People's Hospital in public FDA and regional records.

  128. US regulatory status: approved. Molecular target: Adrenergic receptor alpha-2.

    Target
    Adrenergic receptor alpha-2
    Mechanism
    Adrenergic receptor alpha-2 agonist
  129. clopidogrel

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in First People's Hospital's portfolio. Mechanism: Purinergic receptor P2Y12 antagonist.

    Mechanism
    Purinergic receptor P2Y12 antagonist
  130. Development asset linked to First People's Hospital in public FDA and regional records.

  131. Development asset linked to First People's Hospital in public FDA and regional records.

  132. Development asset linked to First People's Hospital in public FDA and regional records.

  133. Development asset linked to First People's Hospital in public FDA and regional records.

  134. Development asset linked to First People's Hospital in public FDA and regional records.

  135. Development asset linked to First People's Hospital in public FDA and regional records.

  136. Development asset linked to First People's Hospital in public FDA and regional records.

  137. covid-19 vaccine (inactivated, adjuvanted, adsorbed)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in First People's Hospital's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  138. US regulatory status: approved. Molecular target: Complement C5.

    Target
    Complement C5
    Mechanism
    Complement C5 inhibitor
  139. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  140. US regulatory status: approved. Molecular target: Peptidyl-prolyl cis-trans isomerase A.

    Target
    Peptidyl-prolyl cis-trans isomerase A
    Mechanism
    Cyclophilin A modulator
  141. US regulatory status: approved. Molecular target: Cystine.

    Target
    Cystine
    Mechanism
    Cystine reducing agent
  142. cytarabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA polymerase (alpha/delta/epsilon) inhibitor
  143. Development asset linked to First People's Hospital in public FDA and regional records.

  144. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Prothrombin.

    Target
    Prothrombin
    Mechanism
    Thrombin inhibitor
  145. dabigatran etexilate

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in First People's Hospital's portfolio. Mechanism: Thrombin inhibitor.

    Mechanism
    Thrombin inhibitor
  146. dapagliflozin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Sodium/glucose cotransporter 2.

    Target
    Sodium/glucose cotransporter 2
    Mechanism
    Sodium/glucose cotransporter 2 inhibitor
  147. daratumumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1.

    Target
    ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
    Mechanism
    Lymphocyte differentiation antigen CD38 inhibitor
  148. darolutamide

    Antineoplastic and immunomodulating agents (L02)

    US regulatory status: approved. Molecular target: Androgen receptor.

    Target
    Androgen receptor
    Mechanism
    Androgen Receptor antagonist
  149. dasatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Bcr/Abl fusion protein.

    Target
    Bcr/Abl fusion protein
    Mechanism
    SRC inhibitor
  150. decitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA (cytosine-5)-methyltransferase 1.

    Target
    DNA (cytosine-5)-methyltransferase 1
    Mechanism
    DNA (cytosine-5)-methyltransferase 1 inhibitor
  151. Development asset linked to First People's Hospital in public FDA and regional records.

  152. degarelix

    Antineoplastic and immunomodulating agents (L02)

    Antineoplastic and immunomodulating agents (L02) compound in First People's Hospital's portfolio. Mechanism: Gonadotropin-releasing hormone receptor antagonist.

    Mechanism
    Gonadotropin-releasing hormone receptor antagonist
  153. dengue tetravalent vaccine (live, attenuated)

    Antiinfectives for systemic use (J07)

    Antiinfectives for systemic use (J07) compound in First People's Hospital's portfolio. Mechanism: Biological vaccine - induces immune response.

    Mechanism
    Biological vaccine - induces immune response
  154. US regulatory status: approved. Molecular target: Cell membrane.

    Target
    Cell membrane
    Mechanism
    Cell membrane disrupting agent
  155. Development asset linked to First People's Hospital in public FDA and regional records. Mechanism: Vasopressin receptor agonist.

    Mechanism
    Vasopressin receptor agonist
  156. US regulatory status: approved. Molecular target: Vasopressin receptor.

    Target
    Vasopressin receptor
    Mechanism
    Vasopressin receptor agonist
  157. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  158. US regulatory status: approved. Molecular target: Mineralocorticoid receptor.

    Target
    Mineralocorticoid receptor
    Mechanism
    Mineralocorticoid receptor agonist
  159. deucravacitinib

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Non-receptor tyrosine-protein kinase TYK2.

    Target
    Non-receptor tyrosine-protein kinase TYK2
    Mechanism
    Tyrosine-protein kinase TYK2 negative allosteric modulator
  160. US regulatory status: approved. Molecular target: Glucocorticoid receptor.

    Target
    Glucocorticoid receptor
    Mechanism
    Glucocorticoid receptor agonist
  161. Development asset linked to First People's Hospital in public FDA and regional records.

  162. US regulatory status: approved. Molecular target: Potassium-transporting ATPase.

    Target
    Potassium-transporting ATPase
    Mechanism
    Potassium-transporting ATPase inhibitor
  163. dexmedetomidine

    Nervous system (N05)

    Nervous system (N05) compound in First People's Hospital's portfolio. Mechanism: Adrenergic receptor alpha-2 agonist.

    Mechanism
    Adrenergic receptor alpha-2 agonist
  164. US regulatory status: approved. Molecular target: Adrenergic receptor alpha-2.

    Target
    Adrenergic receptor alpha-2
    Mechanism
    Adrenergic receptor alpha-2 agonist
  165. US regulatory status: approved. Molecular target: DNA topoisomerase II.

    Target
    DNA topoisomerase II
    Mechanism
    DNA topoisomerase II inhibitor
  166. US regulatory status: approved. Molecular target: Thyroid hormone receptor.

    Target
    Thyroid hormone receptor
    Mechanism
    Thyroid hormone receptor agonist
  167. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  168. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  169. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  170. Development asset linked to First People's Hospital in public FDA and regional records.

  171. US regulatory status: approved. Molecular target: Sodium/potassium-transporting ATPase.

    Target
    Sodium/potassium-transporting ATPase
    Mechanism
    Sodium/potassium-transporting ATPase inhibitor
  172. US regulatory status: approved. Molecular target: 3',5'-cyclic phosphodiesterase.

    Target
    3',5'-cyclic phosphodiesterase
    Mechanism
    3',5'-cyclic phosphodiesterase inhibitor
  173. Development asset linked to First People's Hospital in public FDA and regional records.

  174. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  175. dolutegravir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved.

  176. Development asset linked to First People's Hospital in public FDA and regional records. Mechanism: Beta-1 adrenergic receptor agonist.

    Mechanism
    Beta-1 adrenergic receptor agonist
  177. dopamine hydrochloride

    Cardiovascular system (C01)

    US regulatory status: approved. Molecular target: Beta-1 adrenergic receptor.

    Target
    Beta-1 adrenergic receptor
    Mechanism
    Beta-1 adrenergic receptor agonist
  178. Development asset linked to First People's Hospital in public FDA and regional records.

  179. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in First People's Hospital's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  180. doxorubicin hydrochloride

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA topoisomerase II alpha inhibitor
  181. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Matrix metalloproteinase-1 inhibitor
  182. US regulatory status: approved. Molecular target: Histamine H1 receptor.

    Target
    Histamine H1 receptor
    Mechanism
    Histamine H1 receptor antagonist
  183. US regulatory status: approved. Molecular target: Mineralocorticoid receptor.

    Target
    Mineralocorticoid receptor
    Mechanism
    Progesterone receptor agonist
  184. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: Fibroblast growth factor receptor 1.

    Target
    Fibroblast growth factor receptor 1
    Mechanism
    Fibroblast growth factor receptor 1 inhibitor
  185. Development asset linked to First People's Hospital in public FDA and regional records.

  186. edaravone

    Nervous system (N07)

    US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  187. Development asset linked to First People's Hospital in public FDA and regional records. Molecular target: IgG receptor FcRn large subunit p51.

    Target
    IgG receptor FcRn large subunit p51
    Mechanism
    IgG receptor FcRn large subunit p51 antagonist
  188. eflornithine

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in First People's Hospital's portfolio. Mechanism: Ornithine decarboxylase inhibitor.

    Mechanism
    Ornithine decarboxylase inhibitor