Friday, July 10, 2026

Drug profile · INN

dipyridamole

dipyridamole (DIPYRIDAMOLE) is a 3',5'-cyclic phosphodiesterase inhibitor. Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 5
Pipeline programs 4
News articles 0
Drug details — dipyridamole
US status
approved
Class
Route
INJECTION
Patents
5
Programs
4
Data quality
0.84

Quick answer

dipyridamole (DIPYRIDAMOLE) is a 3',5'-cyclic phosphodiesterase inhibitor. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN dipyridamole
Brand DIPYRIDAMOLE
Mechanism 3',5'-cyclic phosphodiesterase inhibitor
Target 3',5'-cyclic phosphodiesterase
Route INJECTION
Formulation INJECTABLE

Mechanism of action

3',5'-cyclic phosphodiesterase inhibitor

Primary target: 3',5'-cyclic phosphodiesterase

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. CAMER5UA Phase 3 · United Therapeutics Europe · Cervical Artery Dissection
  2. Dipyridamole 50mg tid Phase 3 · First People's Hospital · Restless Leg Syndrome Due to Uraemia
  3. 114180 Approved · Disc Medicine · Stroke
  4. dipyridamole Approved · United Therapeutics Europe · Coronary Artery Disease

Related & competitor drugs

  1. cilostazol Phosphodiesterase 3A inhibitor
  2. dyphylline Phosphodiesterase 4 inhibitor
  3. sildenafil citrate Phosphodiesterase 5A inhibitor
  4. tadalafil Genito-urinary system and sex hormones (G04)
  5. vardenafil hydrochloride Phosphodiesterase 5A inhibitor
  6. avanafil Genito-urinary system and sex hormones (G04)

Related patents

  1. US 10973758

    Methods of eye treatment using therapeutic compositions containing dipyridamole

    Expires Mon Apr 08 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 10357453

    Methods of eye treatment using therapeutic compositions containing dipyridamole

    Expires Mon Jul 18 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 10322129

    Therapeutic compositions containing dipyridamole, treatment packs and kits including such compositions and methods for producing same

    Expires Mon Jun 13 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 10226420

    Methods of eye treatment using therapeutic compositions containing dipyridamole

    Expires Mon Mar 07 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 9901580

    Methods of eye treatment using therapeutic compositions containing dipyridamole

    Expires Mon Feb 22 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is dipyridamole?

dipyridamole (DIPYRIDAMOLE) is a 3',5'-cyclic phosphodiesterase inhibitor. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for dipyridamole?

DIPYRIDAMOLE is a marketed brand name for dipyridamole. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of dipyridamole?

dipyridamole has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.