Wednesday, June 10, 2026

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Boehringer Ingelheim

Boehringer Ingelheim drug portfolio β€” 113 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Binger Straße, Ingelheim am Rhein, Rhineland-Palatinate 55218, DE HQ
46,699 Employees
NMPA registrant Type
Company details
Status
Public
HQ
Binger Straße, Ingelheim am Rhein, Rhineland-Palatinate 55218, DE
Employees
46,699
Programs
193
Drugs
113
Patents
25
Intelligence Β· Drug Pipeline

Boehringer Ingelheim pipeline

Portfolio lens on 113 drugs and development assets β€” regulatory status, targets, and deep links to NovaPharmaNews drug profiles.

Boehringer Ingelheim drug portfolio β€” 113 indexed compounds with therapeutic class and molecular targets from public FDA and regional approval metadata.

Drug portfolio

113 compounds
  1. afatinib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Mechanism: Epidermal growth factor receptor erbB1 inhibitor.

    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  2. amlodipine

    Cardiovascular system (C09)

    Cardiovascular system (C09) compound in Boehringer Ingelheim's portfolio. Mechanism: Voltage-gated L-type calcium channel blocker.

    Mechanism
    Voltage-gated L-type calcium channel blocker
  3. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  4. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  5. atezolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  6. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  7. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  8. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Molecular target: Hepatitis C virus serine protease, NS3/NS4A.

    Target
    Hepatitis C virus serine protease, NS3/NS4A
    Mechanism
    Hepatitis C virus serine protease, NS3/NS4A inhibitor
  9. bosentan

    Cardiovascular system (C02)

    US regulatory status: approved. Molecular target: Endothelin receptor, ET-A/ET-B.

    Target
    Endothelin receptor, ET-A/ET-B
    Mechanism
    Endothelin receptor, ET-A/ET-B antagonist
  10. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  11. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Dopamine transporter inhibitor.

    Mechanism
    Dopamine transporter inhibitor
  12. caffeine

    Nervous system (N06)

    US regulatory status: approved. Molecular target: Adenosine receptor.

    Target
    Adenosine receptor
    Mechanism
    Adenosine receptor antagonist
  13. US regulatory status: approved.

  14. capecitabine

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  15. US regulatory status: approved. Molecular target: Sodium channel alpha subunit.

    Target
    Sodium channel alpha subunit
    Mechanism
    Sodium channel alpha subunit blocker
  16. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  17. US regulatory status: approved. Mechanism: Unknown.

    Mechanism
    Unknown
  18. cetuximab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Epidermal growth factor receptor.

    Target
    Epidermal growth factor receptor
    Mechanism
    Epidermal growth factor receptor erbB1 inhibitor
  19. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  20. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  21. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  22. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  23. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Molecular target: Prothrombin.

    Target
    Prothrombin
    Mechanism
    Thrombin inhibitor
  24. dabigatran etexilate

    Blood and blood forming organs (B01)

    Blood and blood forming organs (B01) compound in Boehringer Ingelheim's portfolio. Mechanism: Thrombin inhibitor.

    Mechanism
    Thrombin inhibitor
  25. US regulatory status: approved. Molecular target: Sodium/potassium-transporting ATPase.

    Target
    Sodium/potassium-transporting ATPase
    Mechanism
    Sodium/potassium-transporting ATPase inhibitor
  26. docetaxel

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Tubulin.

    Target
    Tubulin
    Mechanism
    Tubulin inhibitor
  27. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  28. doxorubicin

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Boehringer Ingelheim's portfolio. Mechanism: DNA topoisomerase II alpha inhibitor.

    Mechanism
    DNA topoisomerase II alpha inhibitor
  29. durvalumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death 1 ligand 1.

    Target
    Programmed cell death 1 ligand 1
    Mechanism
    Programmed cell death 1 ligand 1 inhibitor
  30. empagliflozin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Sodium/glucose cotransporter 2.

    Target
    Sodium/glucose cotransporter 2
    Mechanism
    Sodium/glucose cotransporter 2 inhibitor
  31. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  32. enoxaparin sodium

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Antithrombin-III.

    Target
    Antithrombin-III
    Mechanism
    Antithrombin-III activator
  33. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  34. US regulatory status: approved. Molecular target: Bacterial 70S ribosome.

    Target
    Bacterial 70S ribosome
    Mechanism
    Bacterial 70S ribosome inhibitor
  35. esomeprazole

    Alimentary tract and metabolism (A02)

    Alimentary tract and metabolism (A02) compound in Boehringer Ingelheim's portfolio. Mechanism: Potassium-transporting ATPase inhibitor.

    Mechanism
    Potassium-transporting ATPase inhibitor
  36. US regulatory status: approved. Molecular target: Estrogen receptor.

    Target
    Estrogen receptor
    Mechanism
    Estrogen receptor alpha agonist
  37. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  38. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    Thymidylate synthase inhibitor
  39. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  40. furosemide

    Cardiovascular system (C03)

    US regulatory status: approved. Molecular target: Solute carrier family 12 member 1.

    Target
    Solute carrier family 12 member 1
    Mechanism
    Sodium-(potassium)-chloride cotransporter 2 inhibitor
  41. glucagon

    Systemic hormonal preparations (H04)

    US regulatory status: approved. Molecular target: Glucagon receptor.

    Target
    Glucagon receptor
    Mechanism
    Glucagon receptor agonist
  42. US regulatory status: approved. Molecular target: Glucagon receptor.

    Target
    Glucagon receptor
    Mechanism
    Glucagon receptor agonist
  43. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  44. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  45. US regulatory status: approved. Molecular target: Enoyl-[acyl-carrier-protein] reductase [NADH] FabI.

    Target
    Enoyl-[acyl-carrier-protein] reductase [NADH] FabI
    Mechanism
    Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor
  46. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  47. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Mu opioid receptor agonist.

    Mechanism
    Mu opioid receptor agonist
  48. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  49. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  50. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  51. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  52. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  53. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  54. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  55. US regulatory status: approved. Molecular target: Lanosterol 14-alpha demethylase.

    Target
    Lanosterol 14-alpha demethylase
    Mechanism
    Cytochrome P450 51 inhibitor
  56. US regulatory status: approved. Molecular target: Cyclooxygenase.

    Target
    Cyclooxygenase
    Mechanism
    Cyclooxygenase inhibitor
  57. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  58. linagliptin

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Dipeptidyl peptidase 4.

    Target
    Dipeptidyl peptidase 4
    Mechanism
    Dipeptidyl peptidase IV inhibitor
  59. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  60. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  61. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Mitochondrial complex I (NADH dehydrogenase) inhibitor.

    Mechanism
    Mitochondrial complex I (NADH dehydrogenase) inhibitor
  62. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Beta-1 adrenergic receptor antagonist.

    Mechanism
    Beta-1 adrenergic receptor antagonist
  63. midazolam

    Nervous system (N05)

    US regulatory status: approved. Molecular target: GABA-A receptor; anion channel.

    Target
    GABA-A receptor; anion channel
    Mechanism
    GABA-A receptor; anion channel positive allosteric modulator
  64. nintedanib

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Mechanism: Vascular endothelial growth factor receptor inhibitor.

    Mechanism
    Vascular endothelial growth factor receptor inhibitor
  65. US regulatory status: approved. Molecular target: Fibroblast growth factor receptor.

    Target
    Fibroblast growth factor receptor
    Mechanism
    Fibroblast growth factor receptor inhibitor
  66. nivolumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  67. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Beta-2 adrenergic receptor agonist.

    Mechanism
    Beta-2 adrenergic receptor agonist
  68. US regulatory status: approved. Molecular target: Potassium-transporting ATPase.

    Target
    Potassium-transporting ATPase
    Mechanism
    Potassium-transporting ATPase inhibitor
  69. US regulatory status: approved. Molecular target: DNA.

    Target
    DNA
    Mechanism
    DNA inhibitor
  70. pembrolizumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Programmed cell death protein 1.

    Target
    Programmed cell death protein 1
    Mechanism
    Programmed cell death protein 1 inhibitor
  71. pemetrexed

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  72. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  73. US regulatory status: approved. Molecular target: Dihydrofolate reductase.

    Target
    Dihydrofolate reductase
    Mechanism
    Thymidylate synthase inhibitor
  74. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  75. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  76. pramipexole

    Nervous system (N04)

    Nervous system (N04) compound in Boehringer Ingelheim's portfolio. Mechanism: D2-like dopamine receptor agonist.

    Mechanism
    D2-like dopamine receptor agonist
  77. US regulatory status: approved. Molecular target: Solute carrier family 22 member 11.

    Target
    Solute carrier family 22 member 11
    Mechanism
    Solute carrier family 22 member 6 inhibitor
  78. repaglinide

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Sulfonylurea receptor 1, Kir6.2.

    Target
    Sulfonylurea receptor 1, Kir6.2
    Mechanism
    Sulfonylurea receptor 1, Kir6.2 blocker
  79. ribavirin

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: Inosine-5'-monophosphate dehydrogenase 1.

    Target
    Inosine-5'-monophosphate dehydrogenase 1
    Mechanism
    Inosine-5'-monophosphate dehydrogenase 1 inhibitor
  80. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: HMG-CoA reductase inhibitor.

    Mechanism
    HMG-CoA reductase inhibitor
  81. semaglutide

    Alimentary tract and metabolism (A10)

    US regulatory status: approved. Molecular target: Glucagon-like peptide 1 receptor.

    Target
    Glucagon-like peptide 1 receptor
    Mechanism
    Glucagon-like peptide 1 receptor agonist
  82. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  83. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  84. spesolimab

    Antineoplastic and immunomodulating agents (L04)

    Antineoplastic and immunomodulating agents (L04) compound in Boehringer Ingelheim's portfolio. Molecular target: IL36 receptor.

    Target
    IL36 receptor
    Mechanism
    IL36 receptor antagonist
  85. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  86. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  87. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  88. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  89. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  90. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  91. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  92. telmisartan

    Cardiovascular system (C09)

    US regulatory status: approved. Molecular target: Type-1 angiotensin II receptor.

    Target
    Type-1 angiotensin II receptor
    Mechanism
    Type-1 angiotensin II receptor antagonist
  93. tenecteplase

    Blood and blood forming organs (B01)

    US regulatory status: approved. Molecular target: Tissue-type plasminogen activator.

    Target
    Tissue-type plasminogen activator
    Mechanism
    Tissue-type plasminogen activator exogenous protein
  94. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  95. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Muscarinic acetylcholine receptor M3 antagonist.

    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  96. US regulatory status: approved. Molecular target: Muscarinic acetylcholine receptor M3.

    Target
    Muscarinic acetylcholine receptor M3
    Mechanism
    Muscarinic acetylcholine receptor M3 antagonist
  97. tipranavir

    Antiinfectives for systemic use (J05)

    US regulatory status: approved. Molecular target: Human immunodeficiency virus type 1 protease.

    Target
    Human immunodeficiency virus type 1 protease
    Mechanism
    Human immunodeficiency virus type 1 protease inhibitor
  98. tocilizumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Interleukin-6 receptor subunit alpha.

    Target
    Interleukin-6 receptor subunit alpha
    Mechanism
    Interleukin-6 receptor alpha subunit inhibitor
  99. trastuzumab

    Antineoplastic and immunomodulating agents (L01)

    US regulatory status: approved. Molecular target: Receptor tyrosine-protein kinase erbB-2.

    Target
    Receptor tyrosine-protein kinase erbB-2
    Mechanism
    Receptor protein-tyrosine kinase erbB-2 inhibitor
  100. trastuzumab deruxtecan

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Boehringer Ingelheim's portfolio. Molecular target: DNA topoisomerase 1.

    Target
    DNA topoisomerase 1
    Mechanism
    DNA topoisomerase I inhibitor
  101. trastuzumab emtansine

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Boehringer Ingelheim's portfolio. Molecular target: Receptor tyrosine-protein kinase erbB-2.

    Target
    Receptor tyrosine-protein kinase erbB-2
    Mechanism
    Tubulin inhibitor
  102. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  103. ustekinumab

    Antineoplastic and immunomodulating agents (L04)

    US regulatory status: approved. Molecular target: Interleukin-12.

    Target
    Interleukin-12
    Mechanism
    Interleukin-23 inhibitor
  104. Development asset linked to Boehringer Ingelheim in public FDA and regional records.

  105. Development asset linked to Boehringer Ingelheim in public FDA and regional records. Mechanism: Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor.

    Mechanism
    Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor
  106. zanidatamab

    Antineoplastic and immunomodulating agents (L01)

    Antineoplastic and immunomodulating agents (L01) compound in Boehringer Ingelheim's portfolio. Molecular target: Receptor tyrosine-protein kinase erbB-2.

    Target
    Receptor tyrosine-protein kinase erbB-2
    Mechanism
    Receptor protein-tyrosine kinase erbB-2 inhibitor