Wednesday, July 8, 2026

Patent intelligence · US

US 9226921

Fused heterocyclic compounds as phosphodiesterases (PDES) inhibitors

granted A61KA61K31/4353A61K31/4355A61K31/437
Status granted
Linked drugs 2
Pipeline programs 6
Years to expiry 9
Applicant portfolio 1,436
Patent details — US 9226921
Jurisdiction
US
Status
granted
Grant date
Jan 5, 2016
Expiration
Dec 31, 2035
Claims
17
CPC classes
A61K, A61K31/4353, A61K31/4355, A61K31/437
View on Google Patents ↗

Quick answer

US 9226921 (Fused heterocyclic compounds as phosphodiesterases (PDES) inhibitors) is held by Takeda Pharmaceutical Company Limited. Status: granted. Granted Jan 5, 2016. Expires Dec 31, 2035 (9 years remaining) — relevant for patent-cliff and LOE planning.

Key facts

Grant date
Expiration
Claims
17
CPC classes
A61K, A61K31/4353, A61K31/4355, A61K31/437, A61K31/4427, A61K31/4439

More from Takeda Pharmaceutical Company Limited

Related pharmaceutical patents in our USPTO index.

  1. US 12428403

    N-(heterocyclyl and heterocyclylalkyl)-3-benzylpyridin-2-amine derivatives as SSTR4 agonists

    Takeda Pharmaceutical Company Limited · Expires Sep 25, 2045

    granted
  2. US 12421188

    Heterocyclic compound and use thereof

    Takeda Pharmaceutical Company Limited · Expires Sep 18, 2045

    granted
  3. US 12419890

    Administration of sumo-activating enzyme inhibitor and checkpoint inhibitors

    Takeda Pharmaceutical Company Limited · Expires Sep 18, 2045

    granted
  4. US 12415866

    Monoclonal antibody inhibitor of Factor XIIa

    Takeda Pharmaceutical Company Limited · Expires Sep 11, 2045

    granted
  5. US 12415782

    Heterocyclic compound and use thereof

    Takeda Pharmaceutical Company Limited · Expires Sep 11, 2045

    granted
  6. US 12409210

    CNS delivery of therapeutic agents

    Takeda Pharmaceutical Company Limited · Expires Sep 4, 2045

    granted
  7. US 12404237

    Method of treating excessive sleepiness and/or cataplexy using n-{2-(([1,1′-biphenyl]-3-yl)methyl)pyrrolidin-3-yl}sulfonamide derivatives

    Takeda Pharmaceutical Company Limited · Expires Aug 28, 2045

    granted
  8. US 12403154

    Administration of sting agonist and checkpoint inhibitors

    Takeda Pharmaceutical Company Limited · Expires Aug 28, 2045

    granted

Frequently asked questions

What is US patent 9226921?

US 9226921 (Fused heterocyclic compounds as phosphodiesterases (PDES) inhibitors) is held by Takeda Pharmaceutical Company Limited. Status: granted. Granted Jan 5, 2016. Expires Dec 31, 2035 (9 years remaining) — relevant for patent-cliff and LOE planning.

Who owns US 9226921?

Takeda Pharmaceutical Company Limited is listed as the applicant in USPTO PatentsView records indexed by NovaPharmaNews. We track 1,436 pharmaceutical patents for this assignee.

When does US 9226921 expire?

Our index shows an expiration date of Dec 31, 2035 (9 years from today). Confirm material dates against USPTO, FDA Orange Book, or qualified counsel before contractual decisions.