Wednesday, July 8, 2026

Drug profile · INN

zilucoplan sodium

zilucoplan sodium (ZILBRYSQ) is a complement c5 binding agent. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved PMDA: approved
US status approved
Patents linked 9
Pipeline programs 3
News articles 0
Drug details — zilucoplan sodium
US status
approved
Class
Route
SUBCUTANEOUS
Patents
9
Programs
3
Data quality
0.84

Quick answer

zilucoplan sodium (ZILBRYSQ) is a complement c5 binding agent. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN zilucoplan sodium
Brand ZILBRYSQ
Mechanism Complement C5 binding agent
Target Complement C5
Route SUBCUTANEOUS
Formulation SOLUTION

Mechanism of action

Complement C5 binding agent

Primary target: Complement C5

Approval history

Authority Status Date
FDA approved
PMDA approved

Pipeline programs

  1. MG0014 Phase 3 · Anaxis Pharma · Generalized Myasthenia Gravis
  2. MG0015 Phase 3 · Anaxis Pharma · Generalized Myasthenia Gravis
  3. Zilucoplan sodium Phase 3 · Anaxis Pharma · Generalized Myasthenia Gravis

Related & competitor drugs

  1. pozelimab-bbfg Complement C5 inhibitor
  2. avacincaptad pegol sodium Complement C5 inhibitor
  3. crovalimab-akkz Complement C5 inhibitor
  4. eculizumab Antineoplastic and immunomodulating agents (L04)
  5. eculizumab-aagh Complement C5 inhibitor
  6. eculizumab-aeeb Complement C5 inhibitor

Related patents

  1. US 11965040

    Modulation of complement activity

    Expires Mon Apr 18 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 11752190

    Modulators of complement activity

    Expires Mon Sep 07 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 11535650

    Modulation of complement activity

    Expires Mon Dec 22 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 11014965

    Modulation of complement activity

    Expires Mon May 20 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 10835574

    Modulators of complement activity

    Expires Mon Nov 12 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 10562934

    Modulation of complement activity

    Expires Mon Feb 13 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. US 10435438

    Modulation of complement activity

    Expires Mon Oct 03 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. US 10208089

    Modulation of complement activity

    Expires Mon Feb 14 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. US 10106579

    Modulation of complement activity

    Expires Mon Oct 18 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is zilucoplan sodium?

zilucoplan sodium (ZILBRYSQ) is a complement c5 binding agent. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for zilucoplan sodium?

ZILBRYSQ is a marketed brand name for zilucoplan sodium. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of zilucoplan sodium?

zilucoplan sodium has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.