Wednesday, July 8, 2026

Drug profile · INN

valbenazine tosylate

valbenazine tosylate (VALBENAZINE TOSYLATE) is a synaptic vesicular amine transporter inhibitor. Associated with NEUROCRINE BIOSCIENCES INC. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 20
Pipeline programs 0
News articles 0
Drug details — valbenazine tosylate
US status
approved
Class
Route
ORAL
Patents
20
Programs
0
Data quality
0.89

Quick answer

valbenazine tosylate (VALBENAZINE TOSYLATE) is a synaptic vesicular amine transporter inhibitor. Associated with NEUROCRINE BIOSCIENCES INC. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN valbenazine tosylate
Brand VALBENAZINE TOSYLATE
Mechanism Synaptic vesicular amine transporter inhibitor
Target Synaptic vesicular amine transporter
Route ORAL
Formulation CAPSULE

Mechanism of action

Synaptic vesicular amine transporter inhibitor

Primary target: Synaptic vesicular amine transporter

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. deutetrabenazine Nervous system (N07)
  2. reserpine Synaptic vesicular amine transporter inhibitor
  3. deserpidine Synaptic vesicular amine transporter inhibitor
  4. rescinnamine Synaptic vesicular amine transporter inhibitor
  5. tetrabenazine Synaptic vesicular amine transporter inhibitor
  6. valbenazine Synaptic vesicular amine transporter inhibitor
  1. US 12421193

    GPR52 modulators and methods of use

    Expires Mon Sep 18 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 11654142

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon May 18 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 11439629

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Sep 08 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 11311532

    High dosage valbenazine formulation and compositions, methods, and kits related thereto

    Expires Mon Apr 21 2042 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 11040029

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Jun 17 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 11026931

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Jun 03 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. US 11026939

    High dosage valbenazine formulation and compositions, methods, and kits related thereto

    Expires Mon Jun 03 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. US 10993941

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Apr 29 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. US 10952997

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Mar 18 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  10. US 10940141

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Mar 04 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  11. US 10912771

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Feb 04 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  12. US 10874648

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Dec 24 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  13. US 10857148

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Dec 03 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  14. US 10857137

    Methods for the administration of certain VMAT2 inhibitors

    Expires Mon Dec 03 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  15. US 10851104

    Valbenazine salts and polymorphs thereof

    Expires Mon Nov 26 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  16. US 10851103

    Valbenazine salts and polymorphs thereof

    Expires Mon Nov 26 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  17. US 10844058

    Valbenazine salts and polymorphs thereof

    Expires Mon Nov 19 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  18. US 10065952

    Valbenazine salts and polymorphs thereof

    Expires Mon Aug 30 2038 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  19. US 8357697

    Substituted 3-isobutyl-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2H-pyrido[2,1-A]isoquinolin-2-ol compounds and methods relating thereto

    Expires Mon Jan 17 2033 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  20. US 8039627

    Substituted 3-isobutyl-9,10-dimethoxy-1,3,4,6,7,11b-hexahydro-2H-pyrido[2,1-A]isoquinolin-2-ol compounds and methods relating thereto

    Expires Mon Oct 13 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is valbenazine tosylate?

valbenazine tosylate (VALBENAZINE TOSYLATE) is a synaptic vesicular amine transporter inhibitor. Associated with NEUROCRINE BIOSCIENCES INC. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for valbenazine tosylate?

VALBENAZINE TOSYLATE is a marketed brand name for valbenazine tosylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of valbenazine tosylate?

valbenazine tosylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.