Saturday, July 11, 2026

Drug profile · INN

upadacitinib hydrate

upadacitinib hydrate (RINVOQ PARTIAL CHANGE APPROVAL) is a tyrosine-protein kinase jak1 inhibitor.

PMDA: approved
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Drug details — upadacitinib hydrate
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Quick answer

upadacitinib hydrate (RINVOQ PARTIAL CHANGE APPROVAL) is a tyrosine-protein kinase jak1 inhibitor.

Key facts

INN upadacitinib hydrate
Brand RINVOQ PARTIAL CHANGE APPROVAL
Mechanism Tyrosine-protein kinase JAK1 inhibitor
Target Tyrosine-protein kinase JAK1

Mechanism of action

Tyrosine-protein kinase JAK1 inhibitor

Primary target: Tyrosine-protein kinase JAK1

Approval history

Authority Status Date
PMDA approved

Related & competitor drugs

  1. abrocitinib Dermatologicals (D11)
  2. baricitinib Antineoplastic and immunomodulating agents (L04)
  3. deuruxolitinib phosphate Tyrosine-protein kinase JAK1 inhibitor
  4. ruxolitinib phosphate Tyrosine-protein kinase JAK2 inhibitor
  5. filgotinib Antineoplastic and immunomodulating agents (L04)
  6. momelotinib Tyrosine-protein kinase JAK1 inhibitor

Frequently asked questions

What is upadacitinib hydrate?

upadacitinib hydrate (RINVOQ PARTIAL CHANGE APPROVAL) is a tyrosine-protein kinase jak1 inhibitor.

What is the brand name for upadacitinib hydrate?

RINVOQ PARTIAL CHANGE APPROVAL is a marketed brand name for upadacitinib hydrate. Check FDA Drugs@FDA for the current US label holder and prescribing information.