Wednesday, July 8, 2026

Drug profile · INN

umbralisib tosylate

umbralisib tosylate (UKONIQ) is a tyrosine-protein kinase abl inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 3
News articles 0
Drug details — umbralisib tosylate
US status
approved
Class
Route
ORAL
Patents
0
Programs
3
Data quality
0.84

Quick answer

umbralisib tosylate (UKONIQ) is a tyrosine-protein kinase abl inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN umbralisib tosylate
Brand UKONIQ
Mechanism Tyrosine-protein kinase ABL inhibitor
Target Casein kinase I isoform epsilon
Route ORAL
Formulation TABLET

Mechanism of action

Tyrosine-protein kinase ABL inhibitor

Primary target: Casein kinase I isoform epsilon

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Umbralisib Phase 2 · TG THERAPEUTICS · Chronic Lymphocytic Leukemia
  2. Umbralisib Phase 2 · TG THERAPEUTICS · Lymphoma
  3. Umbralisib Phase 2 · TG THERAPEUTICS · Marginal Zone Lymphoma

Frequently asked questions

What is umbralisib tosylate?

umbralisib tosylate (UKONIQ) is a tyrosine-protein kinase abl inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for umbralisib tosylate?

UKONIQ is a marketed brand name for umbralisib tosylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of umbralisib tosylate?

umbralisib tosylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.