Saturday, July 11, 2026

Drug profile · INN

trilostane

trilostane (MODRASTANE) is a 3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type ii inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — trilostane
US status
approved
Class
Route
ORAL
Patents
0
Programs
0
Data quality
0.84

Quick answer

trilostane (MODRASTANE) is a 3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type ii inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN trilostane
Brand MODRASTANE
Mechanism 3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type II inhibitor
Target 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2
Route ORAL
Formulation CAPSULE

Mechanism of action

3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type II inhibitor

Primary target: 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2

Approval history

Authority Status Date
FDA approved

Frequently asked questions

What is trilostane?

trilostane (MODRASTANE) is a 3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type ii inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for trilostane?

MODRASTANE is a marketed brand name for trilostane. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of trilostane?

trilostane has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.