Wednesday, July 8, 2026

Drug profile · INN

tolterodine tartrate

tolterodine tartrate (TOLTERODINE TARTRATE) is a muscarinic acetylcholine receptor m2 antagonist. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — tolterodine tartrate
US status
approved
Class
Route
ORAL
Patents
0
Programs
1
Data quality
0.89

Quick answer

tolterodine tartrate (TOLTERODINE TARTRATE) is a muscarinic acetylcholine receptor m2 antagonist. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN tolterodine tartrate
Brand TOLTERODINE TARTRATE
Mechanism Muscarinic acetylcholine receptor M2 antagonist
Target Muscarinic acetylcholine receptor M2
Route ORAL
Formulation CAPSULE, EXTENDED RELEASE

Mechanism of action

Muscarinic acetylcholine receptor M2 antagonist

Primary target: Muscarinic acetylcholine receptor M2

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. doxazosin plus tolterodine SR Approved · Samsung Bioepis · Overactive Bladder

Related & competitor drugs

  1. bethanechol chloride Muscarinic acetylcholine receptor M3 agonist
  2. fesoterodine fumarate Muscarinic acetylcholine receptor M2 antagonist
  3. oxybutynin Genito-urinary system and sex hormones (G04)
  4. oxybutynin chloride Muscarinic acetylcholine receptor M3 antagonist
  5. solifenacin succinate Muscarinic acetylcholine receptor M3 antagonist
  6. darifenacin hydrobromide Genito-urinary system and sex hormones (G04)

Frequently asked questions

What is tolterodine tartrate?

tolterodine tartrate (TOLTERODINE TARTRATE) is a muscarinic acetylcholine receptor m2 antagonist. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for tolterodine tartrate?

TOLTERODINE TARTRATE is a marketed brand name for tolterodine tartrate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of tolterodine tartrate?

tolterodine tartrate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.