Saturday, July 11, 2026

Drug profile · INN

teprotumumab

teprotumumab (TEPEZZA) is a insulin-like growth factor i receptor antagonist.

EMA: approved Antineoplastic and immunomodulating agents (L04) L04AG13
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Drug details — teprotumumab
Class
Antineoplastic and immunomodulating agents (L04)
Route
Patents
0
Programs
0
Data quality
0.83

Quick answer

teprotumumab (TEPEZZA) is a insulin-like growth factor i receptor antagonist.

Key facts

INN teprotumumab
Brand TEPEZZA
Mechanism Insulin-like growth factor I receptor antagonist
Target Insulin-like growth factor 1 receptor
Therapeutic class Antineoplastic and immunomodulating agents (L04)
ATC code L04AG13

Mechanism of action

Insulin-like growth factor I receptor antagonist

Primary target: Insulin-like growth factor 1 receptor

Approval history

Authority Status Date
EMA approved

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is teprotumumab?

teprotumumab (TEPEZZA) is a insulin-like growth factor i receptor antagonist.

What is the brand name for teprotumumab?

TEPEZZA is a marketed brand name for teprotumumab. Check FDA Drugs@FDA for the current US label holder and prescribing information.