Saturday, July 11, 2026

Drug profile · INN

sitagliptin + metformin

sitagliptin + metformin (JANUMET XR) is a dipeptidyl peptidase iv inhibitor. Associated with Alphapharm Pty Ltd.

TGA: approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — sitagliptin + metformin

Quick answer

sitagliptin + metformin (JANUMET XR) is a dipeptidyl peptidase iv inhibitor. Associated with Alphapharm Pty Ltd.

Key facts

INN sitagliptin + metformin
Brand JANUMET XR
Mechanism Dipeptidyl peptidase IV inhibitor
Target Dipeptidyl peptidase 4

Mechanism of action

Dipeptidyl peptidase IV inhibitor

Primary target: Dipeptidyl peptidase 4

Approval history

Authority Status Date
TGA approved

Related & competitor drugs

  1. alogliptin benzoate Alimentary tract and metabolism (A10)
  2. linagliptin Alimentary tract and metabolism (A10)
  3. saxagliptin hydrochloride Dipeptidyl peptidase IV inhibitor
  4. sitagliptin phosphate Dipeptidyl peptidase IV inhibitor
  5. begelomab Antineoplastic and immunomodulating agents (L04)
  6. sitagliptin fumarate Alimentary tract and metabolism (A10)

Frequently asked questions

What is sitagliptin + metformin?

sitagliptin + metformin (JANUMET XR) is a dipeptidyl peptidase iv inhibitor. Associated with Alphapharm Pty Ltd.

What is the brand name for sitagliptin + metformin?

JANUMET XR is a marketed brand name for sitagliptin + metformin. Check FDA Drugs@FDA for the current US label holder and prescribing information.