Wednesday, July 8, 2026

Drug profile · INN

selinexor

selinexor (XPOVIO) is a exportin-1 inhibitor. Associated with Shanghai Antengene Corporation Limited. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved TGA: approved NMPA: clinical trials Antineoplastic and immunomodulating agents (L01) L01XX66
US status approved
Patents linked 20
Pipeline programs 65
News articles 1
Drug details — selinexor
US status
approved
Class
Antineoplastic and immunomodulating agents (L01)
Route
ORAL
Patents
20
Programs
65
Data quality
0.89

Quick answer

selinexor (XPOVIO) is a exportin-1 inhibitor. Associated with Shanghai Antengene Corporation Limited. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN selinexor
Brand XPOVIO
Mechanism Exportin-1 inhibitor
Target Exportin-1
Therapeutic class Antineoplastic and immunomodulating agents (L01)
Route ORAL
Formulation TABLET
ATC code L01XX66

Mechanism of action

Exportin-1 inhibitor

Primary target: Exportin-1

Approval history

Authority Status Date
FDA approved
EMA approved
TGA approved
NMPA clinical trials

Recent coverage

Pipeline programs

  1. M22-574 Phase 3 · AbbVie Deutschland GmbH · Relapsed or Refractory Multiple Myeloma (RRMM)
  2. SELINEXOR for endometrial cancer Phase 3 · Karyopharm Therapeutics · endometrial cancer
  3. Selinexor Phase 3 · Karyopharm Therapeutics · Multiple Myeloma
  4. Selinexor Phase 3 · Karyopharm Therapeutics · Endometrial Cancer
  5. Selinexor Phase 3 · Karyopharm Therapeutics · Dedifferentiated Liposarcoma
  6. Selinexor (combination therapy) Phase 3 · Karyopharm Therapeutics · Relapsed/Refractory Diffuse Large B-cell Lymphoma
  7. XPORT-MF-034 Phase 3 · Karyopharm Therapeutics · Treatment naïve patients with MF
  8. CHOP+selinexor+5-Azacitidine Phase 2 · Chinese Academy of · Peripheral T Cell Lymphoma

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)
  1. US 12371420

    Polymorphs of Selinexor

    Expires Mon Jul 24 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 12291508

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon May 01 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 12076418

    Dually derivatized chitosan nanoparticles and methods of making and using the same for gene transfer in vivo

    Expires Mon Aug 29 2044 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 11807629

    Polymorphs of Selinexor

    Expires Mon Nov 02 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 11787771

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon Oct 12 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 11753401

    Polymorphs of Selinexor

    Expires Mon Sep 07 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. US 11746102

    Polymorphs of selinexor

    Expires Mon Aug 31 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. US 11623011

    Dually derivatized chitosan nanoparticles and methods of making and using the same for gene transfer in vivo

    Expires Mon Apr 06 2043 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. US 11078190

    Polymorphs of selinexor

    Expires Mon Jul 29 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  10. US 11052157

    Enhanced loading of intact, bacterially derived vesicles with small molecule compounds

    Expires Mon Jul 01 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  11. US 11034660

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon Jun 10 2041 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  12. US 10647785

    High concentration chitosan-nucleic acid polyplex compositions

    Expires Mon May 07 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  13. US 10544108

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon Jan 23 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  14. US 10519139

    Polymorphs of Selinexor

    Expires Mon Dec 26 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  15. US 10328159

    Enhanced loading of intact, bacterially derived vesicles with small molecule compounds

    Expires Mon Jun 20 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  16. US 9850323

    High concentration chitosan-nucleic acid polyplex compositions

    Expires Mon Dec 21 2037 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  17. US 9714226

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon Jul 20 2037 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  18. US 9623112

    Dually derivatized chitosan nanoparticles and methods of making and using the same

    Expires Mon Apr 13 2037 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  19. US 9079865

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon Jul 09 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  20. US 8999996

    Hydrazide containing nuclear transport modulators and uses thereof

    Expires Mon Apr 02 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is selinexor?

selinexor (XPOVIO) is a exportin-1 inhibitor. Associated with Shanghai Antengene Corporation Limited. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for selinexor?

XPOVIO is a marketed brand name for selinexor. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of selinexor?

selinexor has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.