Wednesday, July 8, 2026

Drug profile · INN

selexipag

selexipag (UPTRAVI) is a prostanoid ip receptor agonist. Associated with Janssen-Cilag Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved TGA: approved PMDA: approved Blood and blood forming organs (B01) B01AC27
US status approved
Patents linked 1
Pipeline programs 0
News articles 0
Drug details — selexipag
US status
approved
Class
Blood and blood forming organs (B01)
Route
ORAL
Patents
1
Programs
0
Data quality
0.84

Quick answer

selexipag (UPTRAVI) is a prostanoid ip receptor agonist. Associated with Janssen-Cilag Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN selexipag
Brand UPTRAVI
Mechanism Prostanoid IP receptor agonist
Target Prostacyclin receptor
Therapeutic class Blood and blood forming organs (B01)
Route ORAL
Formulation POWDER
ATC code B01AC27

Mechanism of action

Prostanoid IP receptor agonist

Primary target: Prostacyclin receptor

Approval history

Authority Status Date
FDA approved
EMA approved
TGA approved
PMDA approved

Related & competitor drugs

  1. apixaban Blood and blood forming organs (B01)
  2. berotralstat Blood and blood forming organs (B06)
  3. bivalirudin Blood and blood forming organs (B01)
  4. c1 inhibitor (human) Blood and blood forming organs (B06)
  5. clopidogrel Blood and blood forming organs (B01)
  6. dabigatran etexilate Blood and blood forming organs (B01)
  1. US 10188648

    Solid state forms of selexipag

    Expires Mon Jan 24 2039 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is selexipag?

selexipag (UPTRAVI) is a prostanoid ip receptor agonist. Associated with Janssen-Cilag Pty Ltd. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for selexipag?

UPTRAVI is a marketed brand name for selexipag. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of selexipag?

selexipag has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.