Friday, July 10, 2026

Drug profile · INN

saquinavir

saquinavir (FORTOVASE) is a human immunodeficiency virus type 1 protease inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: withdrawn Antiinfectives for systemic use (J05) J05AE01
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — saquinavir
US status
approved
Class
Antiinfectives for systemic use (J05)
Route
ORAL
Patents
0
Programs
0
Data quality
0.84

Quick answer

saquinavir (FORTOVASE) is a human immunodeficiency virus type 1 protease inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN saquinavir
Brand FORTOVASE
Mechanism Human immunodeficiency virus type 1 protease inhibitor
Target Human immunodeficiency virus type 1 protease
Therapeutic class Antiinfectives for systemic use (J05)
Route ORAL
Formulation CAPSULE
ATC code J05AE01

Mechanism of action

Human immunodeficiency virus type 1 protease inhibitor

Primary target: Human immunodeficiency virus type 1 protease

Approval history

Authority Status Date
FDA approved
EMA withdrawn

Related & competitor drugs

  1. atazanavir sulfate Antiinfectives for systemic use (J05)
  2. colistimethate sodium Antiinfectives for systemic use (J01)
  3. covid-19 mrna vaccine Antiinfectives for systemic use (J07)
  4. daptomycin Antiinfectives for systemic use (J01)
  5. darunavir Antiinfectives for systemic use (J05)
  6. dengue tetravalent vaccine (live, attenuated) Antiinfectives for systemic use (J07)

Frequently asked questions

What is saquinavir?

saquinavir (FORTOVASE) is a human immunodeficiency virus type 1 protease inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for saquinavir?

FORTOVASE is a marketed brand name for saquinavir. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of saquinavir?

saquinavir has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.