Wednesday, July 8, 2026

Drug profile · INN

rosiglitazone maleate

rosiglitazone maleate (ROSIGLITAZONE MALEATE) is a peroxisome proliferator-activated receptor gamma agonist. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 2
Pipeline programs 0
News articles 0
Drug details — rosiglitazone maleate
US status
approved
Class
Route
ORAL
Patents
2
Programs
0
Data quality
0.84

Quick answer

rosiglitazone maleate (ROSIGLITAZONE MALEATE) is a peroxisome proliferator-activated receptor gamma agonist. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN rosiglitazone maleate
Brand ROSIGLITAZONE MALEATE
Mechanism Peroxisome proliferator-activated receptor gamma agonist
Target Peroxisome proliferator-activated receptor gamma
Route ORAL
Formulation TABLET

Mechanism of action

Peroxisome proliferator-activated receptor gamma agonist

Primary target: Peroxisome proliferator-activated receptor gamma

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. pioglitazone hydrochloride Peroxisome proliferator-activated receptor gamma agonist
  2. troglitazone Peroxisome proliferator-activated receptor gamma agonist
  3. leriglitazone Alimentary tract and metabolism (A16)
  4. rosiglitazone Alimentary tract and metabolism (A10)

Related patents

  1. US 7632841

    2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate

    Expires Mon Dec 10 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 7435741

    2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate

    Expires Mon Oct 09 2028 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is rosiglitazone maleate?

rosiglitazone maleate (ROSIGLITAZONE MALEATE) is a peroxisome proliferator-activated receptor gamma agonist. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for rosiglitazone maleate?

ROSIGLITAZONE MALEATE is a marketed brand name for rosiglitazone maleate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of rosiglitazone maleate?

rosiglitazone maleate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.