Friday, July 10, 2026

Drug profile · INN

rivastigmine

rivastigmine (EXELON) is a cholinesterases; ache & bche inhibitor. Associated with Novartis Pharmaceuticals. Route of administration: transdermal. Current US regulatory status: approved.

FDA: approved EMA: approved TGA: approved Nervous system (N06) N06DA03
US status approved
Patents linked 2
Pipeline programs 4
News articles 0
Drug details — rivastigmine
US status
approved
Class
Nervous system (N06)
Route
TRANSDERMAL
Patents
2
Programs
4
Data quality
0.89

Quick answer

rivastigmine (EXELON) is a cholinesterases; ache & bche inhibitor. Associated with Novartis Pharmaceuticals. Route of administration: transdermal. Current US regulatory status: approved.

Key facts

INN rivastigmine
Brand EXELON
Mechanism Cholinesterases; ACHE & BCHE inhibitor
Target Cholinesterases; ACHE & BCHE
Therapeutic class Nervous system (N06)
Route TRANSDERMAL
Formulation FILM, EXTENDED RELEASE
ATC code N06DA03

Mechanism of action

Cholinesterases; ACHE & BCHE inhibitor

Primary target: Cholinesterases; ACHE & BCHE

Approval history

Authority Status Date
FDA approved
EMA approved
TGA approved

Pipeline programs

  1. 202000842 Approved · Disc Medicine · Depression
  2. Rivastigmine Approved · Novartis India · Alzheimer's Disease
  3. Rivastigmine transdermal patch Approved · Novartis India · Alzheimer's Disease
  4. rivastigmine patch Unknown · Dong Wang · Alzheimer's Disease

Related & competitor drugs

  1. aripiprazole Nervous system (N05)
  2. brexpiprazole Nervous system (N05)
  3. brivaracetam Nervous system (N03)
  4. bupivacaine Nervous system (N01)
  5. buprenorphine Nervous system (N07)
  6. caffeine citrate Nervous system (N06)
  1. US 2015112285

    Transdermal Therapeutic System For Administering Rivastigmine Or Derivatives Thereof

    Expires Wed Apr 18 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. CA 2785117

    SYSTEME THERAPEUTIQUE TRANSDERMIQUE SERVANT A ADMINISTRER DE LA RIVASTIGMINE OU SES DERIVES

    Expires Wed Jun 25 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is rivastigmine?

rivastigmine (EXELON) is a cholinesterases; ache & bche inhibitor. Associated with Novartis Pharmaceuticals. Route of administration: transdermal. Current US regulatory status: approved.

What is the brand name for rivastigmine?

EXELON is a marketed brand name for rivastigmine. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of rivastigmine?

rivastigmine has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.