Friday, July 10, 2026

Drug profile · INN

rezvilutamide

rezvilutamide is a androgen receptor antagonist.

NMPA: clinical trials
Patents linked 0
Pipeline programs 2
News articles 0
Drug details — rezvilutamide
Class
Route
Patents
0
Programs
2
Data quality
0.70

Quick answer

rezvilutamide is a androgen receptor antagonist.

Key facts

INN rezvilutamide
Mechanism Androgen Receptor antagonist
Target Androgen receptor

Mechanism of action

Androgen Receptor antagonist

Primary target: Androgen receptor

Approval history

Authority Status Date
NMPA clinical trials

Pipeline programs

  1. Rezvilutamide Phase 2 · Chinese Academy of · Metastatic Hormone-Sensitive Prostate Cancer
  2. Rezvilutamide Phase 2 · Zenshine Pharmaceuticals · Prostate Cancer

Related & competitor drugs

  1. bicalutamide Androgen Receptor antagonist
  2. danazol Progesterone receptor agonist
  3. nandrolone decanoate Androgen Receptor agonist
  4. testosterone Genito-urinary system and sex hormones (G03)
  5. testosterone cypionate Androgen Receptor agonist
  6. apalutamide Antineoplastic and immunomodulating agents (L02)

Frequently asked questions

What is rezvilutamide?

rezvilutamide is a androgen receptor antagonist.