Friday, July 10, 2026

Drug profile · INN

remimazolam besylate

remimazolam besylate (BYFAVO) is a gaba-a receptor; anion channel positive allosteric modulator. Route of administration: intravenous. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 10
News articles 0
Drug details — remimazolam besylate
US status
approved
Class
Route
INTRAVENOUS
Patents
0
Programs
10
Data quality
0.84

Quick answer

remimazolam besylate (BYFAVO) is a gaba-a receptor; anion channel positive allosteric modulator. Route of administration: intravenous. Current US regulatory status: approved.

Key facts

INN remimazolam besylate
Brand BYFAVO
Mechanism GABA-A receptor; anion channel positive allosteric modulator
Target GABA-A receptor; anion channel
Route INTRAVENOUS
Formulation POWDER

Mechanism of action

GABA-A receptor; anion channel positive allosteric modulator

Primary target: GABA-A receptor; anion channel

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Remimazolam Besylate Phase 3 · First People's Hospital · Critical Illness; Mechanical Ventilation; Shock
  2. Remimazolam Besylate Phase 3 · Chinese Academy of · Analgesia
  3. Remimazolam besylate Phase 3 · Chinese Academy of · Sedative
  4. Byfavo 20 mg powder for solution for injection Phase 2 · Disc Medicine · stress anxiety, anxiety
  5. Byfavo Approved · Hospital Authority · Bronchoscopy
  6. Remimazolam Besylate for Injection Approved · First People's Hospital · Thoracic Surgery
  7. Remimazolam Unknown · First People's Hospital · Sedation and Analgesia
  8. Remimazolam besylate Unknown · First People's Hospital · Remimazolam

Related & competitor drugs

  1. acamprosate calcium GABA-A receptor; anion channel positive modulator
  2. alprazolam GABA-A receptor; anion channel positive allosteric modulator
  3. butabarbital sodium GABA-A receptor; anion channel positive allosteric modulator
  4. chlordiazepoxide hydrochloride GABA-A receptor; anion channel positive allosteric modulator
  5. clobazam GABA-A receptor; anion channel positive allosteric modulator
  6. clonazepam GABA-A receptor; anion channel positive allosteric modulator

Frequently asked questions

What is remimazolam besylate?

remimazolam besylate (BYFAVO) is a gaba-a receptor; anion channel positive allosteric modulator. Route of administration: intravenous. Current US regulatory status: approved.

What is the brand name for remimazolam besylate?

BYFAVO is a marketed brand name for remimazolam besylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of remimazolam besylate?

remimazolam besylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.