Friday, July 10, 2026

Drug profile · INN

relatlimab

relatlimab (OPDUALAG) is a lymphocyte activation gene 3 protein inhibitor.

EMA: approved Antineoplastic and immunomodulating agents (L01) L01FY02
Patents linked 0
Pipeline programs 13
News articles 3
Drug details — relatlimab

Quick answer

relatlimab (OPDUALAG) is a lymphocyte activation gene 3 protein inhibitor.

Key facts

INN relatlimab
Brand OPDUALAG
Mechanism Lymphocyte activation gene 3 protein inhibitor
Target Lymphocyte activation gene 3 protein
Therapeutic class Antineoplastic and immunomodulating agents (L01)
ATC code L01FY02

Mechanism of action

Lymphocyte activation gene 3 protein inhibitor

Primary target: Lymphocyte activation gene 3 protein

Approval history

Authority Status Date
EMA approved

Recent coverage

Pipeline programs

  1. CA224-047 Phase 3 · Bristol-Myers Squibb Australia · Previously Untreated Metastatic or Unresectable Melanoma
  2. CA224-123 Phase 3 · Bristol-Myers Squibb Australia · Metastatic Colorectal Cancer
  3. CA2241093 Phase 3 · Bristol-Myers Squibb Australia · Non-squamous (NSQ), Stage IV or Recurrent Non-small Cell Lun
  4. CA209-142 Phase 2 · Bristol-Myers Squibb Australia · MSI Negative Colorectal Cancer, MSI Positive Colorectal Canc
  5. CA224-020 Phase 2 · Bristol-Myers Squibb Australia · Neoplasms by site
  6. CA224-048 Phase 2 · Bristol-Myers Squibb Australia · Advanced Malignant Tumors
  7. CA224-104 Phase 2 · Bristol-Myers Squibb Australia · Non small Cell Lung cancer, Non Small Cell Lung Cancer, Non
  8. CA224-1044 Phase 2 · Bristol-Myers Squibb Australia · Melanoma

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is relatlimab?

relatlimab (OPDUALAG) is a lymphocyte activation gene 3 protein inhibitor.

What is the brand name for relatlimab?

OPDUALAG is a marketed brand name for relatlimab. Check FDA Drugs@FDA for the current US label holder and prescribing information.