Saturday, July 11, 2026

Drug profile · INN

regorafenib hydrate

regorafenib hydrate (STIVARGA INITIAL APPROVAL) is a discoidin domain-containing receptor 2 inhibitor.

PMDA: approved
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Drug details — regorafenib hydrate
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Route
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Data quality
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Quick answer

regorafenib hydrate (STIVARGA INITIAL APPROVAL) is a discoidin domain-containing receptor 2 inhibitor.

Key facts

INN regorafenib hydrate
Brand STIVARGA INITIAL APPROVAL
Mechanism Discoidin domain-containing receptor 2 inhibitor
Target Discoidin domain-containing receptor 2

Mechanism of action

Discoidin domain-containing receptor 2 inhibitor

Primary target: Discoidin domain-containing receptor 2

Approval history

Authority Status Date
PMDA approved

Related & competitor drugs

  1. regorafenib Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is regorafenib hydrate?

regorafenib hydrate (STIVARGA INITIAL APPROVAL) is a discoidin domain-containing receptor 2 inhibitor.

What is the brand name for regorafenib hydrate?

STIVARGA INITIAL APPROVAL is a marketed brand name for regorafenib hydrate. Check FDA Drugs@FDA for the current US label holder and prescribing information.