Wednesday, July 8, 2026

Drug profile · INN

rasagiline mesylate

rasagiline mesylate (RASAGILINE MESYLATE) is a monoamine oxidase b inhibitor. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 2
Pipeline programs 9
News articles 0
Drug details — rasagiline mesylate
US status
approved
Class
Route
ORAL
Patents
2
Programs
9
Data quality
0.89

Quick answer

rasagiline mesylate (RASAGILINE MESYLATE) is a monoamine oxidase b inhibitor. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN rasagiline mesylate
Brand RASAGILINE MESYLATE
Mechanism Monoamine oxidase B inhibitor
Target Amine oxidase [flavin-containing] B
Route ORAL
Formulation TABLET

Mechanism of action

Monoamine oxidase B inhibitor

Primary target: Amine oxidase [flavin-containing] B

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Rasagiline Phase 3 · Teva Pharma · Progressive Supranuclear Palsy
  2. rasagiline Phase 3 · Teva Pharma · Restless Legs Syndrome
  3. Rasagiline Phase 2 · Teva Pharma · Dementia
  4. rasagiline mesylate Phase 2 · Teva Pharma · Multiple System Atrophy
  5. Rasagiline Approved · Teva Pharma · Depressive Symptoms
  6. Rasagiline Approved · Teva Pharma · Parkinson's Disease
  7. Rasagiline Approved · Teva Pharma · Sleep Disturbances
  8. Rasagiline Mesylate Approved · Teva Pharma · Parkinson's Disease

Related & competitor drugs

  1. safinamide Nervous system (N04)
  2. safinamide mesylate Monoamine oxidase B inhibitor
  3. selegiline Monoamine oxidase B inhibitor
  4. selegiline hydrochloride Monoamine oxidase B inhibitor
  1. US 7815942

    Rasagiline formulations of improved content uniformity

    Expires Mon Oct 14 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 7572834

    Rasagiline formulations and processes for their preparation

    Expires Mon Aug 06 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is rasagiline mesylate?

rasagiline mesylate (RASAGILINE MESYLATE) is a monoamine oxidase b inhibitor. Associated with Teva Pharma GmbH. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for rasagiline mesylate?

RASAGILINE MESYLATE is a marketed brand name for rasagiline mesylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of rasagiline mesylate?

rasagiline mesylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.