Friday, July 10, 2026

Drug profile · INN

rasagiline

rasagiline (ALZIRAS) is a monoamine oxidase b inhibitor. Associated with Lacuna Pharma Pty Ltd.

EMA: approved TGA: approved NMPA: clinical trials Nervous system (N04) N04BD02
Patents linked 12
Pipeline programs 10
News articles 0
Drug details — rasagiline
Class
Nervous system (N04)
Route
Patents
12
Programs
10
Data quality
0.89

Quick answer

rasagiline (ALZIRAS) is a monoamine oxidase b inhibitor. Associated with Lacuna Pharma Pty Ltd.

Key facts

INN rasagiline
Brand ALZIRAS
Mechanism Monoamine oxidase B inhibitor
Therapeutic class Nervous system (N04)
ATC code N04BD02

Mechanism of action

Monoamine oxidase B inhibitor

Approval history

Authority Status Date
EMA approved
TGA approved
NMPA clinical trials

Pipeline programs

  1. Rasagiline Phase 3 · Teva Pharma · Progressive Supranuclear Palsy
  2. rasagiline Phase 3 · Teva Pharma · Restless Legs Syndrome
  3. Rasagiline Phase 2 · Teva Pharma · Dementia
  4. rasagiline mesylate Phase 2 · Teva Pharma · Multiple System Atrophy
  5. UECHUP-RAS/24-2 Phase 1 · Tillomed Laboratories · Parkinson´s disease
  6. Rasagiline Approved · Teva Pharma · Depressive Symptoms
  7. Rasagiline Approved · Teva Pharma · Parkinson's Disease
  8. Rasagiline Approved · Teva Pharma · Sleep Disturbances

Related & competitor drugs

  1. aripiprazole Nervous system (N05)
  2. brexpiprazole Nervous system (N05)
  3. brivaracetam Nervous system (N03)
  4. bupivacaine Nervous system (N01)
  5. buprenorphine Nervous system (N07)
  6. caffeine citrate Nervous system (N06)
  1. US 12310929

    Use of rasagiline for the treatment of restless legs syndrome

    Expires Mon May 22 2045 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 9308182

    Parenteral formulations of rasagiline

    Expires Mon Apr 07 2036 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 8809310

    Use of rasagiline for the treatment of multiple system atrophy

    Expires Mon Aug 14 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 8691872

    Dispersions of rasagiline citrate

    Expires Mon Apr 03 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  5. US 8569379

    Use of rasagiline for the treatment of olfactory dysfunction

    Expires Mon Oct 24 2033 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  6. US 8080584

    Delayed release rasagiline citrate formulation

    Expires Mon Dec 15 2031 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  7. US 7855233

    Citrate salt of Rasagiline

    Expires Mon Dec 16 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  8. US 7815942

    Rasagiline formulations of improved content uniformity

    Expires Mon Oct 14 2030 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  9. US 7619117

    Rasagiline formulations and processes for their preparation

    Expires Mon Nov 12 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  10. US 7598420

    Rasagiline formulations and processes for their preparation

    Expires Mon Oct 01 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  11. US 7572834

    Rasagiline formulations and processes for their preparation

    Expires Mon Aug 06 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  12. US 7547806

    Tannate salt of rasagiline

    Expires Mon Jun 11 2029 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is rasagiline?

rasagiline (ALZIRAS) is a monoamine oxidase b inhibitor. Associated with Lacuna Pharma Pty Ltd.

What is the brand name for rasagiline?

ALZIRAS is a marketed brand name for rasagiline. Check FDA Drugs@FDA for the current US label holder and prescribing information.