Saturday, July 11, 2026

Drug profile · INN

prilocaine hydrochloride

prilocaine hydrochloride (PRILOCAINE HYDROCHLORIDE) is a sodium channel alpha subunit blocker. Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — prilocaine hydrochloride
US status
approved
Class
Route
INJECTION
Patents
0
Programs
1
Data quality
0.84

Quick answer

prilocaine hydrochloride (PRILOCAINE HYDROCHLORIDE) is a sodium channel alpha subunit blocker. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN prilocaine hydrochloride
Brand PRILOCAINE HYDROCHLORIDE
Mechanism Sodium channel alpha subunit blocker
Target Sodium channel alpha subunit
Route INJECTION
Formulation INJECTABLE

Mechanism of action

Sodium channel alpha subunit blocker

Primary target: Sodium channel alpha subunit

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. PVX 2024-01 Phase 2 · Anaxis Pharma · Subjects having local anesthesia for dental procedures.

Related & competitor drugs

  1. carbamazepine Sodium channel alpha subunit blocker
  2. disopyramide phosphate Sodium channel alpha subunit blocker
  3. eslicarbazepine acetate Nervous system (N03)
  4. fosphenytoin sodium Sodium channel alpha subunit blocker
  5. lacosamide Nervous system (N03)
  6. lamotrigine Sodium channel alpha subunit blocker

Frequently asked questions

What is prilocaine hydrochloride?

prilocaine hydrochloride (PRILOCAINE HYDROCHLORIDE) is a sodium channel alpha subunit blocker. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for prilocaine hydrochloride?

PRILOCAINE HYDROCHLORIDE is a marketed brand name for prilocaine hydrochloride. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of prilocaine hydrochloride?

prilocaine hydrochloride has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.