Friday, July 10, 2026

Drug profile · INN

pioglitazone

pioglitazone (ACTOS) is a peroxisome proliferator-activated receptor gamma agonist. Associated with Alphapharm Pty Ltd.

EMA: approved TGA: approved Alimentary tract and metabolism (A10) A10BD05
Patents linked 0
Pipeline programs 13
News articles 0
Drug details — pioglitazone
Class
Alimentary tract and metabolism (A10)
Route
Patents
0
Programs
13
Data quality
0.89

Quick answer

pioglitazone (ACTOS) is a peroxisome proliferator-activated receptor gamma agonist. Associated with Alphapharm Pty Ltd.

Key facts

INN pioglitazone
Brand ACTOS
Mechanism Peroxisome proliferator-activated receptor gamma agonist
Therapeutic class Alimentary tract and metabolism (A10)
ATC code A10BD05

Mechanism of action

Peroxisome proliferator-activated receptor gamma agonist

Approval history

Authority Status Date
EMA approved
TGA approved

Pipeline programs

  1. CADET-PAD Phase 3 · COLLEGIUM PHARMACEUTICAL · Ischemia of the lower limbs in the course of obstructive art
  2. CLI-06657AA1-03 Phase 3 · Chiesi Farmaceutici S.p.A · Fabry disease (α-galactosidase A deficiency)
  3. D20180102 Phase 3 · PARItec · Vascular calcification and type 1 diabetes
  4. NW-3509/023/III/2024 Phase 3 · Anaxis Pharma · treatment-resistant schizophrenia (TRS)
  5. pioglitazone Phase 3 · HOFFMANN-LA ROCHE · Diabetes Mellitus Type 2
  6. Istaroxime, LActose Phase 2 · WINDTREE THERAPEUTICS INC · Cardiogenic Shock
  7. LTI-03-2001 (RENEW) Phase 2 · Shanghai Zerun Biotechnology · Idiopathic Pulmonary Fibrosis
  8. D9690C00007 Phase 1 · AstraZeneca · Crohn's disease

Related & competitor drugs

  1. agalsidase alfa Alimentary tract and metabolism (A16)
  2. alogliptin Alimentary tract and metabolism (A10)
  3. alogliptin benzoate Alimentary tract and metabolism (A10)
  4. aprepitant Alimentary tract and metabolism (A04)
  5. budesonide Alimentary tract and metabolism (A07)
  6. canagliflozin Alimentary tract and metabolism (A10)

Frequently asked questions

What is pioglitazone?

pioglitazone (ACTOS) is a peroxisome proliferator-activated receptor gamma agonist. Associated with Alphapharm Pty Ltd.

What is the brand name for pioglitazone?

ACTOS is a marketed brand name for pioglitazone. Check FDA Drugs@FDA for the current US label holder and prescribing information.