Friday, July 10, 2026

Drug profile · INN

pilocarpine

pilocarpine (ISOPTO CARPINE) is a muscarinic acetylcholine receptor m3 agonist. Associated with Novartis Pharmaceuticals. Route of administration: ophthalmic. Current US regulatory status: approved.

FDA: approved TGA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — pilocarpine
US status
approved
Class
Route
OPHTHALMIC
Patents
0
Programs
0
Data quality
0.84

Quick answer

pilocarpine (ISOPTO CARPINE) is a muscarinic acetylcholine receptor m3 agonist. Associated with Novartis Pharmaceuticals. Route of administration: ophthalmic. Current US regulatory status: approved.

Key facts

INN pilocarpine
Brand ISOPTO CARPINE
Mechanism Muscarinic acetylcholine receptor M3 agonist
Target Muscarinic acetylcholine receptor M1
Route OPHTHALMIC
Formulation INSERT, EXTENDED RELEASE

Mechanism of action

Muscarinic acetylcholine receptor M3 agonist

Primary target: Muscarinic acetylcholine receptor M1

Approval history

Authority Status Date
FDA approved
TGA approved

Related & competitor drugs

  1. atropine sulfate Sensory organs (S01)
  2. benztropine mesylate Muscarinic acetylcholine receptor M1 antagonist
  3. dicyclomine hydrochloride Muscarinic acetylcholine receptor M3 antagonist
  4. glycopyrrolate Muscarinic acetylcholine receptor M3 antagonist
  5. pilocarpine hydrochloride Muscarinic acetylcholine receptor M3 agonist
  6. scopolamine Muscarinic acetylcholine receptor M1 antagonist

Frequently asked questions

What is pilocarpine?

pilocarpine (ISOPTO CARPINE) is a muscarinic acetylcholine receptor m3 agonist. Associated with Novartis Pharmaceuticals. Route of administration: ophthalmic. Current US regulatory status: approved.

What is the brand name for pilocarpine?

ISOPTO CARPINE is a marketed brand name for pilocarpine. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of pilocarpine?

pilocarpine has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.