Friday, July 10, 2026

Drug profile · INN

pexidartinib

pexidartinib (TURALIO) is a tyrosine-protein kinase receptor flt3 inhibitor.

EMA: refused Antineoplastic and immunomodulating agents (L01) L01XE
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Drug details — pexidartinib
Class
Antineoplastic and immunomodulating agents (L01)
Route
Patents
0
Programs
0
Data quality
0.83

Quick answer

pexidartinib (TURALIO) is a tyrosine-protein kinase receptor flt3 inhibitor.

Key facts

INN pexidartinib
Brand TURALIO
Mechanism Tyrosine-protein kinase receptor FLT3 inhibitor
Target Macrophage colony-stimulating factor 1 receptor
Therapeutic class Antineoplastic and immunomodulating agents (L01)
ATC code L01XE

Mechanism of action

Tyrosine-protein kinase receptor FLT3 inhibitor

Primary target: Macrophage colony-stimulating factor 1 receptor

Approval history

Authority Status Date
EMA refused

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is pexidartinib?

pexidartinib (TURALIO) is a tyrosine-protein kinase receptor flt3 inhibitor.

What is the brand name for pexidartinib?

TURALIO is a marketed brand name for pexidartinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.