Wednesday, July 8, 2026

Drug profile · INN

pexidartinib hydrochloride

pexidartinib hydrochloride (TURALIO) is a tyrosine-protein kinase receptor flt3 inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — pexidartinib hydrochloride
US status
approved
Class
Route
ORAL
Patents
0
Programs
0
Data quality
0.84

Quick answer

pexidartinib hydrochloride (TURALIO) is a tyrosine-protein kinase receptor flt3 inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN pexidartinib hydrochloride
Brand TURALIO
Mechanism Tyrosine-protein kinase receptor FLT3 inhibitor
Target Macrophage colony-stimulating factor 1 receptor
Route ORAL
Formulation CAPSULE

Mechanism of action

Tyrosine-protein kinase receptor FLT3 inhibitor

Primary target: Macrophage colony-stimulating factor 1 receptor

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. sunitinib malate Vascular endothelial growth factor receptor inhibitor
  2. axatilimab-csfr Macrophage colony stimulating factor receptor inhibitor
  3. pexidartinib Antineoplastic and immunomodulating agents (L01)
  4. quizartinib Antineoplastic and immunomodulating agents (L01)
  5. sunitinib Antineoplastic and immunomodulating agents (L01)
  6. axatilimab Macrophage colony stimulating factor receptor inhibitor

Frequently asked questions

What is pexidartinib hydrochloride?

pexidartinib hydrochloride (TURALIO) is a tyrosine-protein kinase receptor flt3 inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for pexidartinib hydrochloride?

TURALIO is a marketed brand name for pexidartinib hydrochloride. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of pexidartinib hydrochloride?

pexidartinib hydrochloride has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.