Friday, July 10, 2026

Drug profile · INN

pegaptanib

pegaptanib (MACUGEN) is a vascular endothelial growth factor a antagonist.

EMA: withdrawn Sensory organs (S01) S01LA03
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — pegaptanib
Class
Sensory organs (S01)
Route
Patents
0
Programs
1
Data quality
0.83

Quick answer

pegaptanib (MACUGEN) is a vascular endothelial growth factor a antagonist.

Key facts

INN pegaptanib
Brand MACUGEN
Mechanism Vascular endothelial growth factor A antagonist
Target Vascular endothelial growth factor A, long form
Therapeutic class Sensory organs (S01)
ATC code S01LA03

Mechanism of action

Vascular endothelial growth factor A antagonist

Primary target: Vascular endothelial growth factor A, long form

Approval history

Authority Status Date
EMA withdrawn

Pipeline programs

  1. pegaptanib sodium Phase 3 · Pfizer · Macular Degeneration

Related & competitor drugs

  1. aflibercept Sensory organs (S01)
  2. atropine sulfate Sensory organs (S01)
  3. bevacizumab Antineoplastic and immunomodulating agents (L01)
  4. bevacizumab-maly Vascular endothelial growth factor A inhibitor
  5. bimatoprost Sensory organs (S01)
  6. atropine Sensory organs (S01)

Frequently asked questions

What is pegaptanib?

pegaptanib (MACUGEN) is a vascular endothelial growth factor a antagonist.

What is the brand name for pegaptanib?

MACUGEN is a marketed brand name for pegaptanib. Check FDA Drugs@FDA for the current US label holder and prescribing information.