Wednesday, July 8, 2026

Drug profile · INN

nintedanib esylate

nintedanib esylate (NINTEDANIB ESYLATE) is a fibroblast growth factor receptor inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 5
News articles 0
Drug details — nintedanib esylate
US status
approved
Class
Route
ORAL
Patents
0
Programs
5
Data quality
0.84

Quick answer

nintedanib esylate (NINTEDANIB ESYLATE) is a fibroblast growth factor receptor inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN nintedanib esylate
Brand NINTEDANIB ESYLATE
Mechanism Fibroblast growth factor receptor inhibitor
Target Fibroblast growth factor receptor
Route ORAL
Formulation CAPSULE

Mechanism of action

Fibroblast growth factor receptor inhibitor

Primary target: Fibroblast growth factor receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. 1199-0378 Phase 3 · Boehringer Ingelheim · Childhood Interstitial Lung Disease
  2. Nintedanib Phase 3 · Boehringer Ingelheim · Idiopathic Pulmonary Fibrosis
  3. Nintedanib Phase 3 · Boehringer Ingelheim · Lung Diseases, Interstitial
  4. APHP220273 Phase 2 · PARItec · Adult patients aged 18 and over with unicentric hyalino-vasc
  5. Nintedanib,Dextromethorphan Phase 2 · First People's Hospital · Idiopathic Pulmonary Fibrosis (IPF)

Related & competitor drugs

  1. pazopanib hydrochloride Vascular endothelial growth factor receptor inhibitor
  2. erdafitinib Antineoplastic and immunomodulating agents (L01)
  3. futibatinib Antineoplastic and immunomodulating agents (L01)
  4. infigratinib phosphate Fibroblast growth factor receptor inhibitor
  5. palifermin Various (V03)
  6. pemigatinib Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is nintedanib esylate?

nintedanib esylate (NINTEDANIB ESYLATE) is a fibroblast growth factor receptor inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for nintedanib esylate?

NINTEDANIB ESYLATE is a marketed brand name for nintedanib esylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of nintedanib esylate?

nintedanib esylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.