Wednesday, July 8, 2026

Drug profile · INN

nilotinib

nilotinib (TASIGNA) is a tyrosine-protein kinase abl inhibitor. Associated with Novartis Pharmaceuticals. Current US regulatory status: approved.

FDA: approved EMA: approved TGA: approved Antineoplastic and immunomodulating agents (L01) L01EA03
US status approved
Patents linked 4
Pipeline programs 11
News articles 2
Drug details — nilotinib

Quick answer

nilotinib (TASIGNA) is a tyrosine-protein kinase abl inhibitor. Associated with Novartis Pharmaceuticals. Current US regulatory status: approved.

Key facts

INN nilotinib
Brand TASIGNA
Mechanism Tyrosine-protein kinase ABL inhibitor
Therapeutic class Antineoplastic and immunomodulating agents (L01)
Formulation CAPSULE
ATC code L01EA03

Mechanism of action

Tyrosine-protein kinase ABL inhibitor

Approval history

Authority Status Date
FDA approved
EMA approved
TGA approved

Recent coverage

Pipeline programs

  1. CABL001A2001B Phase 3 · Novartis India · chronic myelogenous leukemia (CML) or Philadelphia Chromosom
  2. CABL001J12301 Phase 3 · Novartis India · Chronic Myeloid Leukemia
  3. CABL001J12302 Phase 3 · Novartis India · Chronic Myeloid Leukemia
  4. Nilotinib Phase 3 · Novartis India · Chronic Myeloid Leukemia
  5. Nilotinib Phase 3 · Chinese Academy of · Chronic Myeloid Leukemia, Chronic Phase
  6. Nilotinib (AMN107) Phase 3 · Novartis India · Gastrointestinal Stromal Tumor (GIST)
  7. CABL001E2201 Phase 2 · Novartis India · Chronic Myelogenous Leukemia in chronic phase (CML-CP), prev
  8. Nilotinib followed by treatment-free Phase 2 · Novartis India · Chronic Myelogenous Leukemia

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)
  1. US 10640487

    Solid state forms of Nilotinib salts

    Expires Mon Apr 30 2040 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  2. US 9090598

    Nilotinib salts and crystalline forms thereof

    Expires Mon Jul 23 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  3. US 8937082

    Nilotinib salts and crystalline forms thereof

    Expires Mon Jan 15 2035 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted
  4. US 8592442

    Nilotinib HCl crystalline forms

    Expires Mon Nov 21 2033 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is nilotinib?

nilotinib (TASIGNA) is a tyrosine-protein kinase abl inhibitor. Associated with Novartis Pharmaceuticals. Current US regulatory status: approved.

What is the brand name for nilotinib?

TASIGNA is a marketed brand name for nilotinib. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of nilotinib?

nilotinib has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.