Saturday, July 11, 2026

Drug profile · INN

methylergonovine maleate

methylergonovine maleate (METHYLERGONOVINE MALEATE) is a serotonin 2b (5-ht2b) receptor partial agonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — methylergonovine maleate
US status
approved
Class
Route
INJECTION
Patents
0
Programs
0
Data quality
0.89

Quick answer

methylergonovine maleate (METHYLERGONOVINE MALEATE) is a serotonin 2b (5-ht2b) receptor partial agonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: injection. Current US regulatory status: approved.

Key facts

INN methylergonovine maleate
Brand METHYLERGONOVINE MALEATE
Mechanism Serotonin 2b (5-HT2b) receptor partial agonist
Target D(1A) dopamine receptor
Route INJECTION
Formulation INJECTABLE

Mechanism of action

Serotonin 2b (5-HT2b) receptor partial agonist

Primary target: D(1A) dopamine receptor

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. fenoldopam mesylate Dopamine D1 receptor agonist

Frequently asked questions

What is methylergonovine maleate?

methylergonovine maleate (METHYLERGONOVINE MALEATE) is a serotonin 2b (5-ht2b) receptor partial agonist. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: injection. Current US regulatory status: approved.

What is the brand name for methylergonovine maleate?

METHYLERGONOVINE MALEATE is a marketed brand name for methylergonovine maleate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of methylergonovine maleate?

methylergonovine maleate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.