Friday, July 10, 2026

Drug profile · INN

macimorelin

macimorelin (GHRYVELIN (PREVIOUSLY MACIMORELIN AETERNA ZENTARIS)) is a ghrelin receptor agonist.

EMA: approved Various (V04) V04CD06
Patents linked 0
Pipeline programs 0
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Drug details — macimorelin
Class
Various (V04)
Route
Patents
0
Programs
0
Data quality
0.83

Quick answer

macimorelin (GHRYVELIN (PREVIOUSLY MACIMORELIN AETERNA ZENTARIS)) is a ghrelin receptor agonist.

Key facts

INN macimorelin
Brand GHRYVELIN (PREVIOUSLY MACIMORELIN AETERNA ZENTARIS)
Mechanism Ghrelin receptor agonist
Target Growth hormone secretagogue receptor type 1
Therapeutic class Various (V04)
ATC code V04CD06

Mechanism of action

Ghrelin receptor agonist

Primary target: Growth hormone secretagogue receptor type 1

Approval history

Authority Status Date
EMA approved

Related & competitor drugs

  1. besilesomab Various (V09)
  2. deferasirox Various (V03)
  3. ferric citrate coordination complex Various (V03)
  4. folic acid Various (V04)
  5. sevelamer carbonate Various (V03)
  6. sugammadex sodium Various (V03)

Frequently asked questions

What is macimorelin?

macimorelin (GHRYVELIN (PREVIOUSLY MACIMORELIN AETERNA ZENTARIS)) is a ghrelin receptor agonist.

What is the brand name for macimorelin?

GHRYVELIN (PREVIOUSLY MACIMORELIN AETERNA ZENTARIS) is a marketed brand name for macimorelin. Check FDA Drugs@FDA for the current US label holder and prescribing information.