Saturday, July 11, 2026

Drug profile · INN

lomitapide mesylate

lomitapide mesylate (JUXTAPID) is a microsomal triglyceride transfer protein inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — lomitapide mesylate
US status
approved
Class
Route
ORAL
Patents
0
Programs
0
Data quality
0.84

Quick answer

lomitapide mesylate (JUXTAPID) is a microsomal triglyceride transfer protein inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN lomitapide mesylate
Brand JUXTAPID
Mechanism Microsomal triglyceride transfer protein inhibitor
Target Microsomal triglyceride transfer protein
Route ORAL
Formulation CAPSULE

Mechanism of action

Microsomal triglyceride transfer protein inhibitor

Primary target: Microsomal triglyceride transfer protein

Approval history

Authority Status Date
FDA approved

Frequently asked questions

What is lomitapide mesylate?

lomitapide mesylate (JUXTAPID) is a microsomal triglyceride transfer protein inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for lomitapide mesylate?

JUXTAPID is a marketed brand name for lomitapide mesylate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of lomitapide mesylate?

lomitapide mesylate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.