Wednesday, July 8, 2026

Drug profile · INN

lanadelumab-flyo

lanadelumab-flyo (TAKHZYRO) is a plasma kallikrein inhibitor. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 6
News articles 0
Drug details — lanadelumab-flyo
US status
approved
Class
Route
SUBCUTANEOUS
Patents
0
Programs
6
Data quality
0.84

Quick answer

lanadelumab-flyo (TAKHZYRO) is a plasma kallikrein inhibitor. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN lanadelumab-flyo
Brand TAKHZYRO
Mechanism Plasma kallikrein inhibitor
Target Plasma kallikrein
Route SUBCUTANEOUS
Formulation SOLUTION

Mechanism of action

Plasma kallikrein inhibitor

Primary target: Plasma kallikrein

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Lanadelumab Phase 3 · Takeda · Hereditary Angioedema
  2. Lanadelumab Phase 3 · Takeda · Angioedema
  3. Lanadelumab Phase 3 · Takeda · Hereditary Angioedema (HAE)
  4. lanadelumab Phase 2 · Takeda · COVID-19
  5. Lanadelumab Phase 1 · Takeda · COVID-19 Pneumonia
  6. Lanadelumab Phase 1 · Takeda · Healthy Volunteers

Related & competitor drugs

  1. berotralstat dihydrochloride Plasma kallikrein inhibitor
  2. lanadelumab Blood and blood forming organs (B06)
  3. aprotinin Plasminogen inhibitor
  4. ecallantide Plasma kallikrein inhibitor
  5. berotralstat hydrochloride Plasma kallikrein inhibitor

Frequently asked questions

What is lanadelumab-flyo?

lanadelumab-flyo (TAKHZYRO) is a plasma kallikrein inhibitor. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for lanadelumab-flyo?

TAKHZYRO is a marketed brand name for lanadelumab-flyo. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of lanadelumab-flyo?

lanadelumab-flyo has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.