Wednesday, July 8, 2026

Drug profile · INN

icatibant acetate

icatibant acetate (ICATIBANT ACETATE) is a bradykinin b2 receptor antagonist. Associated with Takeda. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 4
News articles 0
Drug details — icatibant acetate
US status
approved
Class
Route
SUBCUTANEOUS
Patents
0
Programs
4
Data quality
0.89

Quick answer

icatibant acetate (ICATIBANT ACETATE) is a bradykinin b2 receptor antagonist. Associated with Takeda. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN icatibant acetate
Brand ICATIBANT ACETATE
Mechanism Bradykinin B2 receptor antagonist
Target B2 bradykinin receptor
Route SUBCUTANEOUS
Formulation INJECTABLE
Originator Takeda

Mechanism of action

Bradykinin B2 receptor antagonist

Primary target: B2 bradykinin receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. Icatibant Phase 3 · Takeda · Angioedema
  2. Icatibant Phase 3 · Takeda · Angiotensin Converting Enzyme Inhibitor Induced Angioedema
  3. Icatibant Phase 3 · Takeda · Hereditary Angioedema
  4. icatibant Phase 3 · Takeda · Hereditary Angioedema (HAE)

Frequently asked questions

What is icatibant acetate?

icatibant acetate (ICATIBANT ACETATE) is a bradykinin b2 receptor antagonist. Associated with Takeda. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for icatibant acetate?

ICATIBANT ACETATE is a marketed brand name for icatibant acetate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of icatibant acetate?

icatibant acetate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.