Saturday, July 11, 2026

Drug profile · INN

esmolol

esmolol is a beta-1 adrenergic receptor antagonist.

NMPA: clinical trials
Patents linked 1
Pipeline programs 1
News articles 0
Drug details — esmolol
Class
Route
Patents
1
Programs
1
Data quality
0.70

Quick answer

esmolol is a beta-1 adrenergic receptor antagonist.

Key facts

INN esmolol
Mechanism Beta-1 adrenergic receptor antagonist

Mechanism of action

Beta-1 adrenergic receptor antagonist

Approval history

Authority Status Date
NMPA clinical trials

Pipeline programs

  1. EUCT 2024-511805-42 Phase 2 · Disc Medicine · Cardiogenic shock

Related patents

  1. AU 2013258031

    Parenteral esmolol formulation

    Expires Wed Nov 15 2034 00:00:00 GMT+0000 (Coordinated Universal Time)

    granted

Frequently asked questions

What is esmolol?

esmolol is a beta-1 adrenergic receptor antagonist.