Friday, July 10, 2026

Drug profile · INN

enfuvirtide

enfuvirtide (FUZEON) is a transmembrane glycoprotein gp41 inhibitor. Route of administration: subcutaneous. Current US regulatory status: approved.

FDA: approved EMA: approved Antiinfectives for systemic use (J05) J05AX07
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — enfuvirtide
US status
approved
Class
Antiinfectives for systemic use (J05)
Route
SUBCUTANEOUS
Patents
0
Programs
0
Data quality
0.84

Quick answer

enfuvirtide (FUZEON) is a transmembrane glycoprotein gp41 inhibitor. Route of administration: subcutaneous. Current US regulatory status: approved.

Key facts

INN enfuvirtide
Brand FUZEON
Mechanism Transmembrane glycoprotein gp41 inhibitor
Target Transmembrane glycoprotein gp41
Therapeutic class Antiinfectives for systemic use (J05)
Route SUBCUTANEOUS
Formulation INJECTABLE
ATC code J05AX07

Mechanism of action

Transmembrane glycoprotein gp41 inhibitor

Primary target: Transmembrane glycoprotein gp41

Approval history

Authority Status Date
FDA approved
EMA approved

Related & competitor drugs

  1. atazanavir sulfate Antiinfectives for systemic use (J05)
  2. colistimethate sodium Antiinfectives for systemic use (J01)
  3. covid-19 mrna vaccine Antiinfectives for systemic use (J07)
  4. daptomycin Antiinfectives for systemic use (J01)
  5. darunavir Antiinfectives for systemic use (J05)
  6. dengue tetravalent vaccine (live, attenuated) Antiinfectives for systemic use (J07)

Frequently asked questions

What is enfuvirtide?

enfuvirtide (FUZEON) is a transmembrane glycoprotein gp41 inhibitor. Route of administration: subcutaneous. Current US regulatory status: approved.

What is the brand name for enfuvirtide?

FUZEON is a marketed brand name for enfuvirtide. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of enfuvirtide?

enfuvirtide has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.