Friday, July 10, 2026

Drug profile · INN

drotrecogin alfa (activated)

drotrecogin alfa (activated) (XIGRIS) is a coagulation factor v inhibitor.

EMA: withdrawn Blood and blood forming organs (B01) B01AD10
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — drotrecogin alfa (activated)
Class
Blood and blood forming organs (B01)
Route
Patents
0
Programs
1
Data quality
0.83

Quick answer

drotrecogin alfa (activated) (XIGRIS) is a coagulation factor v inhibitor.

Key facts

INN drotrecogin alfa (activated)
Brand XIGRIS
Mechanism Coagulation factor V inhibitor
Target Coagulation factor V
Therapeutic class Blood and blood forming organs (B01)
ATC code B01AD10

Mechanism of action

Coagulation factor V inhibitor

Primary target: Coagulation factor V

Approval history

Authority Status Date
EMA withdrawn

Pipeline programs

  1. Drotrecogin alfa (activated) Phase 3 · Eli Lilly and · Sepsis

Related & competitor drugs

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  4. c1 inhibitor (human) Blood and blood forming organs (B06)
  5. clopidogrel Blood and blood forming organs (B01)
  6. dabigatran etexilate Blood and blood forming organs (B01)

Frequently asked questions

What is drotrecogin alfa (activated)?

drotrecogin alfa (activated) (XIGRIS) is a coagulation factor v inhibitor.

What is the brand name for drotrecogin alfa (activated)?

XIGRIS is a marketed brand name for drotrecogin alfa (activated). Check FDA Drugs@FDA for the current US label holder and prescribing information.