Wednesday, July 8, 2026

Drug profile · INN

dorzolamide hydrochloride

dorzolamide hydrochloride (DORZOLAMIDE HYDROCHLORIDE AND TIMOLOL MALEATE) is a carbonic anhydrase ii inhibitor. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: ophthalmic. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 0
News articles 0
Drug details — dorzolamide hydrochloride
US status
approved
Class
Route
OPHTHALMIC
Patents
0
Programs
0
Data quality
0.89

Quick answer

dorzolamide hydrochloride (DORZOLAMIDE HYDROCHLORIDE AND TIMOLOL MALEATE) is a carbonic anhydrase ii inhibitor. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: ophthalmic. Current US regulatory status: approved.

Key facts

INN dorzolamide hydrochloride
Brand DORZOLAMIDE HYDROCHLORIDE AND TIMOLOL MALEATE
Mechanism Carbonic anhydrase II inhibitor
Target Carbonic anhydrase 2
Route OPHTHALMIC
Formulation SOLUTION/DROPS

Mechanism of action

Carbonic anhydrase II inhibitor

Primary target: Carbonic anhydrase 2

Approval history

Authority Status Date
FDA approved

Related & competitor drugs

  1. topiramate GABA-A receptor; anion channel positive modulator
  2. brinzolamide Sensory organs (S01)

Frequently asked questions

What is dorzolamide hydrochloride?

dorzolamide hydrochloride (DORZOLAMIDE HYDROCHLORIDE AND TIMOLOL MALEATE) is a carbonic anhydrase ii inhibitor. Associated with Regeneron Ireland Designated Activity Company (DAC). Route of administration: ophthalmic. Current US regulatory status: approved.

What is the brand name for dorzolamide hydrochloride?

DORZOLAMIDE HYDROCHLORIDE AND TIMOLOL MALEATE is a marketed brand name for dorzolamide hydrochloride. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of dorzolamide hydrochloride?

dorzolamide hydrochloride has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.