Friday, July 10, 2026

Drug profile · INN

dabrafenib mesilate

dabrafenib mesilate (TAFINLAR INITIAL APPROVAL) is a serine/threonine-protein kinase b-raf inhibitor.

PMDA: approved
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Drug details — dabrafenib mesilate
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Quick answer

dabrafenib mesilate (TAFINLAR INITIAL APPROVAL) is a serine/threonine-protein kinase b-raf inhibitor.

Key facts

INN dabrafenib mesilate
Brand TAFINLAR INITIAL APPROVAL
Mechanism Serine/threonine-protein kinase B-raf inhibitor
Target Serine/threonine-protein kinase B-raf

Mechanism of action

Serine/threonine-protein kinase B-raf inhibitor

Primary target: Serine/threonine-protein kinase B-raf

Approval history

Authority Status Date
PMDA approved

Related & competitor drugs

  1. dabrafenib mesylate Serine/threonine-protein kinase B-raf inhibitor
  2. encorafenib Antineoplastic and immunomodulating agents (L01)
  3. vemurafenib Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is dabrafenib mesilate?

dabrafenib mesilate (TAFINLAR INITIAL APPROVAL) is a serine/threonine-protein kinase b-raf inhibitor.

What is the brand name for dabrafenib mesilate?

TAFINLAR INITIAL APPROVAL is a marketed brand name for dabrafenib mesilate. Check FDA Drugs@FDA for the current US label holder and prescribing information.