Friday, July 10, 2026

Drug profile · INN

cyclizine lactate

cyclizine lactate (MAREZINE) is a histamine h1 receptor antagonist. Route of administration: injection. Current US regulatory status: approved.

FDA: approved
US status approved
Patents linked 0
Pipeline programs 1
News articles 0
Drug details — cyclizine lactate
US status
approved
Class
Route
INJECTION
Patents
0
Programs
1
Data quality
0.84

Quick answer

cyclizine lactate (MAREZINE) is a histamine h1 receptor antagonist. Route of administration: injection. Current US regulatory status: approved.

Key facts

INN cyclizine lactate
Brand MAREZINE
Mechanism Histamine H1 receptor antagonist
Target Histamine H1 receptor
Route INJECTION
Formulation INJECTABLE

Mechanism of action

Histamine H1 receptor antagonist

Primary target: Histamine H1 receptor

Approval history

Authority Status Date
FDA approved

Pipeline programs

  1. D8460C00004 Phase 2 · AstraZeneca · Investigating obesity or overweight condition correlated to

Related & competitor drugs

  1. azelastine hydrochloride Histamine H1 receptor antagonist
  2. brompheniramine maleate Histamine H1 receptor antagonist
  3. carbinoxamine maleate Histamine H1 receptor antagonist
  4. cetirizine hydrochloride Histamine H1 receptor antagonist
  5. chlorpheniramine maleate Histamine H1 receptor antagonist
  6. clemastine fumarate Histamine H1 receptor antagonist

Frequently asked questions

What is cyclizine lactate?

cyclizine lactate (MAREZINE) is a histamine h1 receptor antagonist. Route of administration: injection. Current US regulatory status: approved.

What is the brand name for cyclizine lactate?

MAREZINE is a marketed brand name for cyclizine lactate. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of cyclizine lactate?

cyclizine lactate has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.