Friday, July 10, 2026

Drug profile · INN

cenerimod

cenerimod is a sphingosine 1-phosphate receptor edg-1 modulator.

NMPA: clinical trials
Patents linked 0
Pipeline programs 5
News articles 0
Drug details — cenerimod
Class
Route
Patents
0
Programs
5
Data quality
0.70

Quick answer

cenerimod is a sphingosine 1-phosphate receptor edg-1 modulator.

Key facts

INN cenerimod
Mechanism Sphingosine 1-phosphate receptor Edg-1 modulator
Target Sphingosine 1-phosphate receptor 1

Mechanism of action

Sphingosine 1-phosphate receptor Edg-1 modulator

Primary target: Sphingosine 1-phosphate receptor 1

Approval history

Authority Status Date
NMPA clinical trials

Pipeline programs

  1. Cenerimod Phase 3 · Viatris Pharmaceuticals Co · Lupus Erythematosus, Systemic
  2. Cenerimod 4 mg Phase 3 · Viatris Pharmaceuticals Co · Systemic lupus erythematosus
  3. Cenerimod 4 mg, Cenerimod matching placebo Phase 3 · Viatris Pharmaceuticals Co · Moderate to severe systemic lupus erythematosus
  4. Cenerimod matching placebo, Cenerimod 4 mg Phase 3 · Viatris Pharmaceuticals Co · Moderate to severe systemic lupus erythematosus
  5. ID-064-108 Phase 1 · Viatris Pharmaceuticals Co · Not applicable - healthy volunteer trial

Related & competitor drugs

  1. ponesimod Antineoplastic and immunomodulating agents (L04)
  2. etrasimod arginine Sphingosine 1-phosphate receptor Edg-6 modulator
  3. ozanimod hydrochloride Sphingosine 1-phosphate receptor Edg-1 modulator
  4. siponimod Antineoplastic and immunomodulating agents (L04)
  5. etrasimod Antineoplastic and immunomodulating agents (L04)
  6. siponimod fumaric acid Sphingosine 1-phosphate receptor Edg-1 agonist

Frequently asked questions

What is cenerimod?

cenerimod is a sphingosine 1-phosphate receptor edg-1 modulator.