Wednesday, July 8, 2026

Drug profile · INN

cedazuridine

cedazuridine (INAQOVI) is a cytidine deaminase inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved Antineoplastic and immunomodulating agents (L01) L01BC58
US status approved
Patents linked 0
Pipeline programs 3
News articles 0
Drug details — cedazuridine
US status
approved
Class
Antineoplastic and immunomodulating agents (L01)
Route
ORAL
Patents
0
Programs
3
Data quality
0.84

Quick answer

cedazuridine (INAQOVI) is a cytidine deaminase inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN cedazuridine
Brand INAQOVI
Mechanism Cytidine deaminase inhibitor
Target Cytidine deaminase
Therapeutic class Antineoplastic and immunomodulating agents (L01)
Route ORAL
Formulation TABLET
ATC code L01BC58

Mechanism of action

Cytidine deaminase inhibitor

Primary target: Cytidine deaminase

Approval history

Authority Status Date
FDA approved
EMA approved

Pipeline programs

  1. ASTX030-01 Phase 3 · Taiho Pharma Canada · Myelodysplastic Syndromes (MDS), Chronic Myelomonocytic Leuk
  2. ASTX727-17 Phase 1 · Taiho Pharma Canada · Acute myeloid lymphoma (AML), myelodysplastic syndrome (MDS)
  3. ASTX727-18 Phase 1 · Taiho Pharma Canada · Solid tumor, Acute myeloid lymphoma (AML), Myelodysplastic s

Related & competitor drugs

  1. abiraterone acetate Antineoplastic and immunomodulating agents (L02)
  2. anagrelide Antineoplastic and immunomodulating agents (L01)
  3. apremilast Antineoplastic and immunomodulating agents (L04)
  4. arsenic trioxide Antineoplastic and immunomodulating agents (L01)
  5. axitinib Antineoplastic and immunomodulating agents (L01)
  6. azacitidine Antineoplastic and immunomodulating agents (L01)

Frequently asked questions

What is cedazuridine?

cedazuridine (INAQOVI) is a cytidine deaminase inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for cedazuridine?

INAQOVI is a marketed brand name for cedazuridine. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of cedazuridine?

cedazuridine has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.