Wednesday, July 8, 2026

Drug profile · INN

brensocatib

brensocatib (BRINSUPRI) is a dipeptidyl peptidase i inhibitor. Route of administration: oral. Current US regulatory status: approved.

FDA: approved EMA: approved Respiratory system (R03) R03
US status approved
Patents linked 0
Pipeline programs 2
News articles 0
Drug details — brensocatib
US status
approved
Class
Respiratory system (R03)
Route
ORAL
Patents
0
Programs
2
Data quality
0.84

Quick answer

brensocatib (BRINSUPRI) is a dipeptidyl peptidase i inhibitor. Route of administration: oral. Current US regulatory status: approved.

Key facts

INN brensocatib
Brand BRINSUPRI
Mechanism Dipeptidyl peptidase I inhibitor
Target Dipeptidyl peptidase 1
Therapeutic class Respiratory system (R03)
Route ORAL
Formulation TABLET
ATC code R03

Mechanism of action

Dipeptidyl peptidase I inhibitor

Primary target: Dipeptidyl peptidase 1

Approval history

Authority Status Date
FDA approved
EMA approved

Pipeline programs

  1. INS1007-231 Phase 2 · Insmed Incorporated · Hidradenitis Suppurativa
  2. The BiRCh Study Phase 2 · Insmed Incorporated · Chronic Rhinosinusitis without Nasal Polyps (CRSsNP)

Related & competitor drugs

  1. desloratadine Respiratory system (R01)
  2. deutivacaftor / tezacaftor / vanzacaftor Respiratory system (R07)
  3. ivacaftor Respiratory system (R07)
  4. lumacaftor Respiratory system (R07)
  5. mannitol Respiratory system (R05)
  6. reslizumab Respiratory system (R03)

Frequently asked questions

What is brensocatib?

brensocatib (BRINSUPRI) is a dipeptidyl peptidase i inhibitor. Route of administration: oral. Current US regulatory status: approved.

What is the brand name for brensocatib?

BRINSUPRI is a marketed brand name for brensocatib. Check FDA Drugs@FDA for the current US label holder and prescribing information.

What is the US approval status of brensocatib?

brensocatib has approved status in the United States according to our Drugs@FDA-derived records. Verify on the official FDA label before clinical or commercial decisions.